SCHEMBL8764124

SCHEMBL8764124

C=CCOC(=O)C(Br)C(=O)C(N)CC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 10/20 0.34
MAPT P10636 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
GRIK1 P39086 2/20 0.31
GRIK2 Q13002 2/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 2/20 0.30
ALDH1A1 P00352 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
BLM P54132 1/20 0.30
SLC6A3 Q01959 1/20 0.30
MEN1 O00255 1/20 0.30
CYP2D6 P10635 1/20 0.30
NFKB1 P19838 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532116 0.83 MAPT (0.38) CASP1MAPTCACNA1BAPBA1GRIK1
SCHEMBL1023366 0.83 MAPT (0.38) CASP1MAPTCACNA1BAPBA1GRIK1
Hydrochloric Acid SCHEMBL8140432 0.81 MAPT (0.37) CASP1MAPTCACNA1BAPBA1GRIK1
SCHEMBL27566951 0.80 SMN1; SMN2 (0.36) TSHRTDP1CYP2D6
SCHEMBL27546128 0.71 TDP1 (0.35) CASP1MAPTCACNA1BAPBA1CYP3A4
SCHEMBL6745057 0.70 CASP1 (0.35) CASP1MAPTCACNA1BAPBA1GRIK1
SCHEMBL27587694 0.70 TDP1 (0.38) CASP1MAPTCACNA1BAPBA1CYP3A4
SCHEMBL2524519 0.70 TDP1 (0.40) MAPTCACNA1BAPBA1CYP3A4TSHR
SCHEMBL367991 0.70 SMN1; SMN2 (0.44) CASP1MAPTCACNA1BAPBA1CYP3A4
SCHEMBL7489183 0.70 SMN1; SMN2 (0.44) CASP1MAPTCACNA1BAPBA1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed