SCHEMBL8764759

SCHEMBL8764759

C=CCOC(=O)NC(CC(=O)COC(=O)c1c(Cl)cccc1Cl)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 17/20 0.47
ITGB2 P05107 1/20 0.42
ICAM1 P05362 1/20 0.42
ITGAL P20701 1/20 0.42
TXNRD1 Q16881 1/20 0.42
CASP3 P42574 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6801048 0.79 CASP3 (0.52) CASP1ITGB2ICAM1ITGALTXNRD1
SCHEMBL13178975 0.78 CASP1 (0.48) CASP1CASP3
SCHEMBL644624 0.78 CASP1 (0.48) CASP1CASP3
SCHEMBL645654 0.78 CASP1 (0.48) CASP1CASP3
SCHEMBL6281724 0.77 CASP1 (0.59) CASP1CASP3
SCHEMBL6801541 0.77 CASP1 (0.59) CASP1CASP3
SCHEMBL7256039 0.76 CASP1 (0.50) CASP1CASP3
SCHEMBL6800767 0.76 RECQL (0.52) ITGB2ICAM1ITGALCASP3
SCHEMBL646188 0.75 CASP1 (0.44) CASP1CASP3
SCHEMBL4439353 0.75 CYP3A4 (0.58) TXNRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed