SCHEMBL8765147

SCHEMBL8765147

CC(=O)Nc1ccc(-c2c(C(F)F)nn(-c3ccc(NC(C)=O)cc3)c2-c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.48
PTGS2 P35354 4/20 0.41
POLB P06746 2/20 0.41
HTT P42858 1/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
GFER P55789 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
EPHX2 P34913 2/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766177 0.96 AOC3 (0.46) AOC3PTGS2POLBHTTEPHX2
SCHEMBL8765030 0.95 POLB (0.48) AOC3PTGS2POLBHTTEPHX2
SCHEMBL8764387 0.91 CA1 (0.51) PTGS2CA12CA1CA2CA9
SCHEMBL8765507 0.88 PTGS2 (0.43) PTGS2
SCHEMBL8765313 0.87 PTGS2 (0.48) PTGS2POLBHTTCA12CA1
SCHEMBL8765550 0.87 PTGS2 (0.46) AOC3PTGS2
SCHEMBL8764490 0.86 CA1 (0.48) PTGS2POLBHTTCA12CA1
SCHEMBL8764467 0.85 CCR1 (0.43) AOC3PTGS2MAPT
SCHEMBL8765491 0.85 PTGS2 (0.47) AOC3PTGS2KDM4EMAPT
SCHEMBL8765351 0.83 PTGS2 (0.43) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-B1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1997-08-06 EP disclosed
US-5639777-A 1,4,5-triphenyl pyrazolyl compounds for the treatment of inflammation and inflammation-related disorders G.D. SEARLE & CO. (US) 1997-06-17 US disclosed
US-5401765-A FOR TREATING ARTHRITIS, PAIN AND FEVER Searle, G. D. (US) 1995-03-28 US disclosed