SCHEMBL8765333

SCHEMBL8765333

CCCC(O)C1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CPN1 P15169 1/20 0.37
CPB2 Q96IY4 1/20 0.37
GPR4 P46093 1/20 0.35
KCNH2 Q12809 1/20 0.35
GNAI3 P08754 5/20 0.34
GNAO1 P09471 5/20 0.34
GNAI1 P63096 5/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24073205 0.88 KCNH2 (0.35) CPN1CPB2KCNH2
SCHEMBL7333024 0.88 GAA (0.41) GNAI3GNAO1GNAI1
SCHEMBL13153397 0.88 KCNH2 (0.35) CPN1CPB2KCNH2
SCHEMBL9435793 0.86 GNAI3 (0.42) GNAI3GNAO1GNAI1
SCHEMBL7876684 0.84
SCHEMBL28892 0.82 CPN1 (0.39) CPN1CPB2GPR4KCNH2GNAI3
SCHEMBL6371560 0.80 CPN1 (0.38) CPN1CPB2GPR4KCNH2SLC6A2
SCHEMBL22066364 0.79 CPN1 (0.41) CPN1CPB2SLC6A2SLC6A4SLC6A3
SCHEMBL11892780 0.79 TP53 (0.50)
SCHEMBL6370619 0.79 CPN1 (0.41) CPN1CPB2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625509-B1 N-alkyl substituted piperidine-derivatives with neurokinin receptor antagonist activity ZENECA LTD (GB) 1997-07-30 EP disclosed
US-5521199-A TREATMENT OF ASTHMA ZENECA LIMITED (GB) 1996-05-28 US disclosed
EP-0625509-A1 N-alkyl substituted piperidine-derivatives with neurokinin receptor antagonist activity ZENECA LIMITED (GB) 1994-11-23 EP disclosed