SCHEMBL8766258

SCHEMBL8766258

CCCc1ccc(-c2cc(F)c(C#Cc3ccc(F)c(F)c3)c(F)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
RARB P10826 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
RARA P10276 1/20 0.36
RARG P13631 1/20 0.36
TP53 P04637 1/20 0.36
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TSHR P16473 1/20 0.36
GRM5 P41594 1/20 0.35
ACACB O00763 3/20 0.34
MCL1 Q07820 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8767540 0.92 TSHR (0.43) CYP17A1CYP11B1CYP11B2RARBHSD17B10
SCHEMBL8766681 0.91 HSD17B10 (0.49) RARBHSD17B10RARARARGTP53
SCHEMBL9512422 0.90 HSD17B10 (0.41) CYP17A1CYP11B1CYP11B2RARBHSD17B10
SCHEMBL8766844 0.90 HSD17B10 (0.51) RARBHSD17B10RAB9ARARARARG
SCHEMBL8767207 0.90 HSD17B10 (0.51) RARBHSD17B10RAB9ARARARARG
SCHEMBL8766246 0.89 CYP17A1 (0.39) CYP17A1CYP11B1CYP11B2RARBRARA
SCHEMBL9434002 0.88 RARB (0.34) RARBHSD17B10NPC1RAB9ARARA
SCHEMBL8755364 0.87 CYP17A1 (0.38) CYP17A1CYP11B1CYP11B2RARBHSD17B10
SCHEMBL25548582 0.86 FFAR1 (0.42) RARBHSD17B10NPC1RAB9ARARA
SCHEMBL8767559 0.86 TSHR (0.41) CYP11B1CYP11B2HSD17B10TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543244-B1 Fluoro substituted tolans and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 1997-08-20 EP disclosed
US-5372746-A Fluoro-substituted tolane compounds and liquid crystalline mixtures containing same HOFFMANN-LA ROCHE INC. (US) 1994-12-13 US disclosed
EP-0543244-A1 Fluoro substituted tolans and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed