SCHEMBL8766246

SCHEMBL8766246

CCc1ccc(-c2cc(F)c(C#Cc3ccc(F)c(F)c3)c(F)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
GRM5 P41594 1/20 0.37
CYP2A6 P11509 1/20 0.36
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ACACB O00763 1/20 0.31
PIK3CA P42336 4/20 0.31
MTOR P42345 4/20 0.31
TRPV3 Q8NET8 1/20 0.31
FAAH O00519 1/20 0.31
GCGR P47871 1/20 0.31
MAPK14 Q16539 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9508806 0.89 GRM5 (0.41) CYP17A1CYP11B1CYP11B2GRM5CYP2A6
SCHEMBL8766258 0.89 CYP17A1 (0.37) CYP17A1CYP11B1CYP11B2GRM5RARA
SCHEMBL8767540 0.86 TSHR (0.43) CYP17A1CYP11B1CYP11B2GRM5RARA
SCHEMBL8766681 0.85 HSD17B10 (0.49) RARARARBRARGMEN1KMT2A
SCHEMBL8755905 0.84 CYP2A6 (0.40) CYP2A6RARARARBRARGACACB
SCHEMBL12736435 0.84 CYP2A6 (0.45) GRM5CYP2A6RARARARBRARG
SCHEMBL8767207 0.84 HSD17B10 (0.51) RARARARBRARGMEN1KMT2A
SCHEMBL8766844 0.84 HSD17B10 (0.51) RARARARBRARGMEN1KMT2A
SCHEMBL8767150 0.83 CHRNA7 (0.41) CYP11B1CYP11B2GRM5L3MBTL1
SCHEMBL8979061 0.82 CYP2A6 (0.44) CYP2A6ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543244-B1 Fluoro substituted tolans and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 1997-08-20 EP disclosed
US-5372746-A Fluoro-substituted tolane compounds and liquid crystalline mixtures containing same HOFFMANN-LA ROCHE INC. (US) 1994-12-13 US disclosed
EP-0543244-A1 Fluoro substituted tolans and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed