SCHEMBL8766259

SCHEMBL8766259

Cc1ccc(N(c2ccc(C)cc2)c2cc(C)cc(N(c3ccc(C)cc3)c3ccc(C)cc3)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
TSHR P16473 1/20 0.48
ACHE P22303 5/20 0.42
TDP1 Q9NUW8 2/20 0.42
MAPT P10636 2/20 0.35
CYP2C19 P33261 2/20 0.35
MCOLN3 Q8TDD5 1/20 0.35
CA2 P00918 2/20 0.35
LPL P06858 1/20 0.35
LIPG Q9Y5X9 1/20 0.35
CYP1A2 P05177 3/20 0.33
CYP2A6 P11509 2/20 0.33
RAPGEF4 Q8WZA2 2/20 0.33
APP P05067 1/20 0.33
CA1 P00915 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL883713 0.95 ALDH1A1 (0.48) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL1108690 0.95 ALDH1A1 (0.48) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL313428 0.95 ALDH1A1 (0.52) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL16153694 0.89 ALDH1A1 (0.40) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL14732550 0.88 ALDH1A1 (0.42) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL13929900 0.88 ALDH1A1 (0.42) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL14732554 0.88 ALDH1A1 (0.42) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL14732552 0.88 ALDH1A1 (0.42) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL2439851 0.87 ALDH1A1 (0.46) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL997789 0.87 ALDH1A1 (0.46) ALDH1A1TSHRACHETDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3345983-B1 COMPOUNDS CONTAINING AT LEAST ONE DISILYL COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS, DISILYLDIBENZOTHIOPHENES, DISILYLDIBENZOPHOSPHOLES, DISILYLDIBENZOTHIOPHENE S-OXIDES AND DISILYLDIBENZOTHIOPHENE S, S-DIOXIDES UDC IRELAND LTD (IE) 2020-08-26 EP disclosed
EP-3457452-A2 OLED DISPLAY WITH EXTENDED LIFETIME UDC Ireland Limited (IE) 2019-03-20 EP disclosed
EP-3345983-A1 COMPOUNDS CONTAINING AT LEAST ONE DISILYL COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS, DISILYLDIBENZOTHIOPHENES, DISILYLDIBENZOPHOSPHOLES, DISILYLDIBENZOTHIOPHENE S-OXIDES AND DISILYLDIBENZOTHIOPHENE S, S-DIOXIDES UDC Ireland Limited (IE) 2018-07-11 EP disclosed
EP-2173834-B1 ORGANIC LIGHT-EMITTING DIODES COMPRISING AT LEAST ONE DISILYL COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS and DISILYLDIBENZOTHIOPHENES UDC IRELAND LTD (IE) 2018-02-14 EP disclosed
US-8981354-B2 Organic light-emitting polymer and device CAMBRIDGE DISPLAY TECHNOLOGY LIMITED (GB) 2015-03-17 US disclosed
US-20130146852-A1 ORGANIC LIGHT-EMITTING POLYMER AND DEVICE SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-06-13 US disclosed
US-8373159-B2 Organic light-emitting diodes comprising carbene-transition metal complex emitter, and at least one compound selected from disilylcarbazoles, disilyldibenzofurans, disilyldibenzothiophenes, disilyldibenzophospholes, disilyldibenzothiophene s-oxides and disilyldibe BASF SE (DE) 2013-02-12 US disclosed
US-8373159-B2 Organic light-emitting diodes comprising carbene-transition metal complex emitter, and at least one compound selected from disilylcarbazoles, disilyldibenzofurans, disilyldibenzothiophenes, disilyldibenzophospholes, disilyldibenzothiophene s-oxides and disilyldibe BASF SE (DE) 2013-02-12 US disclosed
US-8241764-B2 OLED display with extended lifetime BASF AKTIENGESELLSCHAFT (DE) 2012-08-14 US disclosed
US-8241764-B2 OLED display with extended lifetime BASF AKTIENGESELLSCHAFT (DE) 2012-08-14 US disclosed
WO-2009003919-A1 ORGANIC LIGHT-EMITTING DIODES COMPRISING AT LEAST ONE DISILYL COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS, DISILYLDIBENZOTHIOPHENES, DISILYLDIBENZOPHOSPHOLES, DISILYLDIBENZOTHIOPHENE S-OXIDES AND DISILYLDIBENZOTHIOPHENE S,S-DIOXIDES BASF SE (DE) 2009-01-08 WO disclosed
WO-2009003898-A1 ORGANIC LIGHT-EMITTING DIODES CONTAINING CARBENE TRANSITION METAL COMPLEX EMITTERS AND AT LEAST ONE COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS, DISILYLDIBENZOTHIOPHENES, DISILYLDIBENZOPHOSPHOLES, DISILYLDIBENZOTHIOPHENE S-OXIDES AND DISILYLDIBENZOTHIOPHENE S,S-DIOXIDES BASF SE (DE) 2009-01-08 WO disclosed
WO-2008034758-A2 OLED DISPLAY WITH EXTENDED LIFETIME BASF SE (DE) 2008-03-27 WO disclosed
EP-0420207-B1 Electrophotosensitive material and method of manufacturing the same MITA INDUSTRIAL CO LTD (JP) 1997-08-13 EP disclosed
EP-0390196-B1 Electrophotosensitive material MITA INDUSTRIAL CO LTD (JP) 1995-09-20 EP disclosed
US-5185228-A Binder resin, charge transfer material; stability MITA INDUSTRIAL CO., LTD. (JP) 1993-02-09 US disclosed
US-5128229-A Polycarbonate, m-phenylenediamine derivative MITA INDUSTRIAL CO., LTD. (JP) 1992-07-07 US disclosed
US-5059503-A Used for copying machine MITA INDUSTRIAL CO., LTD. (JP) 1991-10-22 US disclosed
EP-0413338-A1 Electrophotosensitive material MITA INDUSTRIAL CO. LTD. (JP) 1991-02-20 EP disclosed
EP-0390196-A2 Electrophotosensitive material MITA INDUSTRIAL CO., LTD. (JP) 1990-10-03 EP disclosed