SCHEMBL8766277

SCHEMBL8766277

C[SiH](C)Oc1c(/C=C/c2ccc(C(=O)O)cc2)ccc(C(C)(C)C)c1C1(C)CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARB P10826 17/20 0.40
RARG P13631 17/20 0.40
RARA P10276 15/20 0.40
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
BLM P54132 1/20 0.34
CASP7 P55210 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
RXRA P19793 3/20 0.31
NR2E1 Q9Y466 1/20 0.31
XDH P47989 1/20 0.31
TNFRSF1A P19438 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766298 1.00 RARB (0.40) RARBRARGRARATP53CYP3A4
SCHEMBL9078557 0.89 ALDH1A1 (0.35) RARBRARGRARACYP3A4MAPT
SCHEMBL9317947 0.82 RARB (0.48) RARBRARGRARATP53CYP3A4
SCHEMBL8766212 0.82 RARB (0.48) RARBRARGRARATP53CYP3A4
SCHEMBL8766203 0.82 RARB (0.48) RARBRARGRARATP53CYP3A4
SCHEMBL8766160 0.81 RARA (0.46) RARBRARGRARATP53CYP3A4
SCHEMBL8766140 0.81 RARA (0.46) RARBRARGRARATP53CYP3A4
SCHEMBL8766895 0.81
SCHEMBL9077144 0.80 RARA (0.33) RARBRARGRARA
SCHEMBL9077961 0.72 RARB (0.38) RARBRARGRARACYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0584191-B1 NOVEL AROMATIC AND POLYCYCLIC COMPOUNDS AND THEIR USE IN HUMAN OR VETERINARY MEDICINE AND IN COSMETICS CIRD GALDERMA (FR) 1997-08-13 EP disclosed
EP-0584191-A1 NOVEL AROMATIC AND POLYCYCLIC COMPOUNDS AND THEIR USE IN HUMAN OR VETERINARY MEDECINE AND IN COSMETICS. CIRD GALDERMA (FR) 1994-03-02 EP disclosed
WO-1992019583-A1 NOVEL AROMATIC AND POLYCYCLIC COMPOUNDS AND THEIR USE IN HUMAN OR VETERINARY MEDECINE AND IN COSMETICS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (CIRD GALDERMA) (FR) 1992-11-12 WO disclosed