SCHEMBL8766916

SCHEMBL8766916

CC/C(=C(\c1ccc(I)cc1)c1ccc(OCCCCN2CCCC2)cc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 13/20 1.00
PDE1B Q01064 13/20 1.00
PDE1C Q14123 13/20 1.00
ESR1 P03372 6/20 0.88
ESR2 Q92731 1/20 0.88
PSMB1 P20618 3/20 0.77
PSMB5 P28074 2/20 0.77
PSMB2 P49721 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8767419 0.98 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL8767418 0.98 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL8767423 0.98 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
Idoxifene SCHEMBL19217 0.93 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
Idoxifene SCHEMBL19216 0.93 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
Idoxifene SCHEMBL3774574 0.93 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL23266947 0.92 ESR1 (0.90) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL7650153 0.87 PSMB1 (1.00) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL30902018 0.87 PSMB1 (1.00) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL29822053 0.87 PSMB1 (1.00) PDE1APDE1BPDE1CESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0638064-B1 SUBSTITUTED 1,1,2-TRIPHENYLBUTENES AND THEIR USE IN THE TREATMENT AND DIAGNOSIS OF CANCER BRITISH TECH GROUP (GB) 1997-08-13 EP disclosed
US-5589500-A TREATMENT OF TUMORS OR ANTICARCINOGENIC AGENTS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1996-12-31 US disclosed
WO-1993022275-A1 SUBSTITUTED 1,1,2-TRIPHENYLBUTENES AND THEIR USE IN THE TREATMENT AND DIAGNOSIS OF CANCER BRITISH TECHNOLOGY GROUP LTD (GB) 1993-11-11 WO disclosed