SCHEMBL8767706

SCHEMBL8767706

NC(N)=NC(=O)c1ccc(Oc2ccc(F)cc2)c(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 18/20 0.53
CYP2C9 P11712 9/20 0.53
CYP2C19 P33261 8/20 0.53
CYP3A4 P08684 6/20 0.53
ADRA1D P25100 1/20 0.47
HTR2A P28223 1/20 0.47
SLC6A3 Q01959 1/20 0.47
SLC9A2 Q9UBY0 1/20 0.47
CYP2D6 P10635 3/20 0.46
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8505886 0.99 SLC9A1 (0.52) SLC9A1CYP2C9CYP2C19CYP3A4ADRA1D
Hydrochloric Acid SCHEMBL8506601 0.88 SLC9A1 (0.52) SLC9A1CYP2C9CYP2C19CYP3A4ADRA1D
Hydrochloric Acid SCHEMBL8503964 0.88 SLC9A1 (0.49) SLC9A1CYP2C9CYP2C19CYP3A4ADRA1D
SCHEMBL27352800 0.85 PARP10 (0.42) SLC9A1CYP2C9CYP2C19CYP3A4
SCHEMBL8181857 0.83 SLC9A1 (0.41) SLC9A1CYP2C9CYP2C19CYP3A4ADRA1D
Hydrochloric Acid SCHEMBL8070333 0.82 SLC9A1 (0.43) SLC9A1CYP2C9CYP2C19CYP3A4ADRA1D
SCHEMBL8641351 0.81 EPAS1 (0.45) SLC9A1CYP2C9CYP2C19CYP3A4SLC9A2
SCHEMBL8185434 0.80 SLC9A1 (0.52) SLC9A1CYP2C9CYP2C19CYP3A4ADRA1D
SCHEMBL8169938 0.80 SLC9A1 (0.39) SLC9A1CYP2C9CYP2C19CYP3A4ADRA1D
Hydrochloric Acid SCHEMBL8640823 0.79 BACE1 (0.46) SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612723-B1 Substituted benzoylguanidines, process for their preparation, their use as medicament, as inhibitor of the cellular Na+/H+ exchange or as diagnostic agent and medicament containing them HOECHST AG (DE) 1997-08-27 EP claimed