SCHEMBL8185434

SCHEMBL8185434

NC(N)=NC(=O)c1ccc(Oc2cccnc2)c(C(F)(F)F)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 9/20 0.52
CYP2C9 P11712 5/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
CYP2C19 P33261 5/20 0.45
CYP2D6 P10635 3/20 0.45
CYP3A4 P08684 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 1/20 0.41
TNF P01375 1/20 0.41
RAB9A P51151 1/20 0.41
NOD1 Q9Y239 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ADRA1D P25100 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8183089 0.91 SMN1; SMN2 (0.47) SLC9A1CYP2C9SMN1; SMN2CYP2C19CYP2D6
SCHEMBL27436629 0.87 SMN1; SMN2 (0.51) SLC9A1CYP2C9SMN1; SMN2KDM4EMEN1
Hydrochloric Acid SCHEMBL8503964 0.85 SLC9A1 (0.49) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL8170154 0.84 SMN1; SMN2 (0.46) SLC9A1CYP2C9SMN1; SMN2KDM4EMEN1
SCHEMBL8004583 0.81 AOC3 (0.49) SMN1; SMN2
SCHEMBL7995072 0.81 ALDH1A1 (0.53) SMN1; SMN2CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL8831863 0.81 SMN1; SMN2 (0.49) SMN1; SMN2KDM4EMEN1ALDH1A1GAA
SCHEMBL8767706 0.80 SLC9A1 (0.53) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL8104657 0.80 AOC3 (0.50) SMN1; SMN2
SCHEMBL8207485 0.80 ALDH1A1 (0.57) SMN1; SMN2KDM4EMEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022883-A Heterocyclyloxybenzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-02-08 US disclosed
US-5665739-A CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-09-09 US disclosed
EP-0694537-A1 Heterocyclyloxy- benzoylguanidine derivatives, their preparation and their use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GmbH (DE) 1996-01-31 EP disclosed