SCHEMBL8768684

SCHEMBL8768684

COc1ccc(C(=O)C(O)OC(O)C(=O)c2ccc(OC)c(Cl)c2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 7/20 0.50
TAS1R1 Q7RTX1 7/20 0.50
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
KMT2A Q03164 4/20 0.46
MAPT P10636 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MEN1 O00255 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HTT P42858 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
KCNH2 Q12809 1/20 0.46
TP53 P04637 1/20 0.46
CYP2D6 P10635 1/20 0.46
ALOX15 P16050 1/20 0.46
LMNA P02545 2/20 0.45
TTR P02766 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9222707 0.83 TAS1R3 (0.52) TAS1R3TAS1R1NPC1RAB9AKMT2A
SCHEMBL12514129 0.83 TAS1R3 (0.57) TAS1R3TAS1R1NPC1RAB9AKMT2A
SCHEMBL8638562 0.82 TAS1R3 (0.51) TAS1R3TAS1R1NPC1RAB9AKMT2A
Hydrochloric Acid SCHEMBL9836181 0.79 TAS1R3 (0.52) TAS1R3TAS1R1NPC1RAB9AKMT2A
SCHEMBL11575925 0.79 CYP1A2 (0.68) TAS1R3TAS1R1NPC1RAB9AKMT2A
SCHEMBL23792352 0.78 TAS1R3 (0.51) TAS1R3TAS1R1NPC1RAB9AKMT2A
SCHEMBL8767461 0.78 HSP90AA1 (0.46) SMN1; SMN2LMNATSHRKDM4ETHRB
SCHEMBL311716 0.78 ADRB2 (0.60) TAS1R3TAS1R1NPC1RAB9AKMT2A
SCHEMBL30446783 0.78 TAS1R3 (0.52) TAS1R3TAS1R1NPC1RAB9AKMT2A
SCHEMBL29524334 0.78 TPMT (0.69) TAS1R3TAS1R1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579833-B1 ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY FUJISAWA PHARMACEUTICAL CO (JP) 1997-08-20 EP disclosed
EP-0579833-A1 ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY. FUJISAWA PHARMACEUTICAL CO (JP) 1994-01-26 EP disclosed
WO-1992018461-A1 ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-10-29 WO disclosed