SCHEMBL8768870

SCHEMBL8768870

CCCCCCCN(C(=O)NCc1ccc(OC(C)(C)C(=O)OCC)cc1)c1ccccc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 10/20 0.44
PPARG P37231 4/20 0.44
HDAC1 Q13547 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
ABCB11 O95342 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
HTR2A P28223 1/20 0.40
PMP22 Q01453 1/20 0.40
PPARD Q03181 3/20 0.39
ADAMTS5 Q9UNA0 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
LTB4R2 Q9NPC1 2/20 0.37
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9111447 0.91 PPARA (0.47) PPARAPPARGHDAC1HDAC6PPARD
SCHEMBL8768939 0.87 PPARA (0.45) PPARAPPARGHDAC1HDAC6ABCB11
SCHEMBL8768894 0.83 PPARA (0.50) PPARAPPARGHDAC1HDAC6ABCB11
SCHEMBL8767770 0.80 PPARA (0.47) PPARAPPARGHDAC1HDAC6ABCB11
SCHEMBL8768867 0.78 PPARA (0.48) PPARAPPARGHDAC1HDAC6ABCB11
SCHEMBL8924428 0.75 PPARA (0.42) PPARAPPARGABCB11CYP1A2CYP3A4
SCHEMBL8768094 0.74 PPARA (0.56) PPARAPPARGABCB11CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11449524 0.72 PPARA (0.58) PPARAPPARGABCB11CYP1A2CYP3A4
SCHEMBL8769015 0.70 PPARA (0.49) PPARAPPARGHDAC1HDAC6ABCB11
SCHEMBL11449966 0.69 PPARA (0.57) PPARAPPARGABCB11CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639178-B1 ANTI-ATHEROSCLEROTIC ARYL COMPOUNDS WELLCOME FOUND (GB) 1997-09-03 EP disclosed
US-5658944-A ANTICHOLESTEROL AGENTS THE UNIVERSITY OF SOUTH CAROLINA (US) 1997-08-19 US disclosed