SCHEMBL8769880

SCHEMBL8769880

O=C1CN(C[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C(=O)N1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.57
CTSL P07711 9/20 0.46
CTSB P07858 8/20 0.46
CTSS P25774 2/20 0.46
CTSK P43235 2/20 0.46
TACR1 P25103 2/20 0.44
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.44
MAPK1 P28482 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
CYP3A4 P08684 1/20 0.43
TRPM8 Q7Z2W7 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ALOX15 P16050 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4202065 0.79 CTRB1 (0.62) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL7361852 0.77 CTRB1 (0.64) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL7361850 0.77 CTRB1 (0.64) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL26745215 0.76 GAA (0.55) NPC1GAAMAPK1RAB9ASMN1; SMN2
SCHEMBL2435512 0.75 CTRB1 (0.76) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL2482903 0.75 CTRB1 (0.76) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL1051352 0.75 CTRB1 (0.76) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL7398976 0.74 CTRB1 (0.60) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL7398974 0.74 CTRB1 (0.60) CTRB1CTSLCTSBCTSSCTSK
SCHEMBL14069202 0.74 CTRB1 (0.60) CTRB1CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793673-A1 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR Takeda Chemical Industries, Ltd. (JP) 1997-09-10 EP disclosed
WO-1996016079-A2 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1996-05-30 WO disclosed