SCHEMBL87699

SCHEMBL87699

C=CC=CC=Cc1ccccc1.C=CCOC(=O)C=C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
CYP3A4 P08684 1/20 0.44
THRB P10828 1/20 0.43
CASP1 P29466 1/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
APP P05067 1/20 0.42
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.40
HSD17B10 Q99714 2/20 0.40
ALOX12 P18054 1/20 0.40
MAOB P27338 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HDAC3 O15379 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11073729 0.88 THRB (0.48) LMNAMEN1KMT2AKDM4EGAA
SCHEMBL10747808 0.88 LMNA (0.42) LMNAMEN1KMT2AKDM4EGAA
Juarezic Acid SCHEMBL203895 0.87 HDAC3 (0.45) LMNAMEN1KMT2AKDM4EGAA
Acrylic Acid Ethyl Ester SCHEMBL580632 0.86 LMNA (0.49) LMNAMEN1KMT2AKDM4EGAA
SCHEMBL170861 0.85 LMNA (0.42) LMNAMEN1KMT2AKDM4EGAA
SCHEMBL7625573 0.84 TSHR (0.53) LMNAMEN1KMT2ACYP3A4THRB
SCHEMBL7265789 0.84 APP (0.51) LMNAMEN1KMT2AKDM4EGAA
Acrylic Acid SCHEMBL2060241 0.83 APP (0.48) LMNAMEN1KMT2AKDM4EGAA
SCHEMBL28152774 0.82 CYP3A4 (0.46) LMNAMEN1KMT2AKDM4EGAA
SCHEMBL87755 0.82 LMNA (0.47) LMNAMEN1KMT2AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2199 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4119598-A1 NANOCOMPOSITE MATERIALS COMPRISING MECHANICAL LIGANDS Nanocore ApS (DK) 2023-01-18 EP claimed
US-20210230381-A1 DESIGN OF COMPOSITE MATERIALS WITH DESIRED CHARACTERISTICS NANOCORE APS (DK) 2021-07-29 US claimed
US-20200291579-A1 COMPOSITE STRUCTURES FOR PACKAGING ARTICLES AND RELATED METHODS SMART PLANET TECHNOLOGIES, INC. 2020-09-17 US claimed
EP-3481891-B1 EXPANDABLE COMPOSITIONS CONTAINING AROMATIC VINYL POLYMERS HAVING SELF-EXTINGUISHING PROPERTIES AND IMPROVED PROCESSABILITY VERSALIS SPA (IT) 2020-04-08 EP claimed
US-20190144622-A1 EXPANDABLE COMPOSITIONS CONTAINING AROMATIC VINYL POLYMERS HAVING SELF-EXTINGUISHING PROPERTIES AND IMPROVED PROCESSABILITY VERSALIS S.P.A. (IT) 2019-05-16 US claimed
EP-3481891-A1 EXPANDABLE COMPOSITIONS CONTAINING AROMATIC VINYL POLYMERS HAVING SELF-EXTINGUISHING PROPERTIES AND IMPROVED PROCESSABILITY Versalis S.p.A. (IT) 2019-05-15 EP claimed
CN-109415527-A Expandable compositions comprising aromatic vinyl polymers having self-extinguishing properties and improved processability 维尔萨利斯股份公司 2019-03-01 CN claimed
WO-2018007602-A1 EXPANDABLE COMPOSITIONS CONTAINING AROMATIC VINYL POLYMERS HAVING SELF-EXTINGUISHING PROPERTIES AND IMPROVED PROCESSABILITY VERSALIS S.P.A. (IT) 2018-01-11 WO claimed
EP-1259565-B1 SILICA REINFORCED RUBBER COMPOSITIONS OF IMPROVED PROCESSABILITY AND STORAGE STABILITY PIRELLI (IT) 2008-11-26 EP claimed
US-6822037-B2 BLENDS CONTAINING SILICA AND ELASTOMER; TIRES; MELT PROCESSABILITY, STORAGE STABILITY PIRELLI PNEUMATICI S.P.A. (IT) 2004-11-23 US claimed
US-6737466-B2 INCREASING CURE RATE BY INCLUDING AN EPOXY COMPOUND, AN ABIETYL COMPOUND, STYRENATED RESORCINOL FORMALDEHYDE EPOXY POLYMER COMPOUND, OR AN ESTER HYDROXYL COMPOUND OF A MOLECULAR WEIGHT BELOW 7,000 PIRELLI PNEUMATICI S.P.A. (IT) 2004-05-18 US claimed
US-20030187110-A1 Silica reinforced rubber compositions of improved processability and storage stability PIRELLI PNEUMATICI S.P.A. (IT) 2003-10-02 US claimed
US-20030158317-A1 Silica reinforced rubber compositions of improved processability and storage stability PIRELLI PNEUMATICI S.P.A. (IT) 2003-08-21 US claimed
EP-1259565-A1 SILICA REINFORCED RUBBER COMPOSITIONS OF IMPROVED PROCESSABILITY AND STORAGE STABILITY PIRELLI PNEUMATICI S.p.A. (IT) 2002-11-27 EP claimed
US-6482884-B1 Silica reinforced rubber compositions of improved processability and storage stability PIRELLI PNEUMATICI S.P.A. (IT) 2002-11-19 US claimed
WO-2001064782-B1 SILICA REINFORCED RUBBER COMPOSITIONS OF IMPROVED PROCESSABILITY AND STORAGE STABILITY PIRELLI (IT) 2002-02-14 WO claimed
WO-2001064782-A1 SILICA REINFORCED RUBBER COMPOSITIONS OF IMPROVED PROCESSABILITY AND STORAGE STABILITY PIRELLI PNEUMATICI S.P.A. (IT) 2001-09-07 WO claimed
US-6391949-B1 None US disclosed
US-4810740-A ACRYLONITRILE-BUTADIENE-STYRENE TERPOLYMER, A METHYLENEDIPHENOL CIBA-GEIGY CORPORATION (US) 1989-03-07 US disclosed
US-4429039-A SUBBING LAYER CONTAINING AN ADDITION COPOLYMER AND A DICHLORO-2-TRIAZINE DERIVATIVE FUJI PHOTO FILM CO., LTD. (JP) 1984-01-31 US disclosed