SCHEMBL8771439

SCHEMBL8771439

CCN(CC)CCNC(=O)c1cc(Cl)ccc1N

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.67
KDM4E B2RXH2 2/20 0.67
HPGD P15428 1/20 0.67
LMNA P02545 3/20 0.59
SLC22A1 O15245 2/20 0.59
CYP1A2 P05177 2/20 0.59
ADRA2A P08913 2/20 0.59
CYP2D6 P10635 2/20 0.59
DRD3 P35462 2/20 0.59
HTR3E A5X5Y0 1/20 0.59
HTR3B O95264 1/20 0.59
MPO P05164 1/20 0.59
DRD2 P14416 1/20 0.59
ADRA2C P18825 1/20 0.59
DRD4 P21917 1/20 0.59
HTR2A P28223 1/20 0.59
HTR2C P28335 1/20 0.59
HTR2B P41595 1/20 0.59
HTR3A P46098 1/20 0.59
KCNH2 Q12809 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8771566 0.92 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDLMNASLC22A1
SCHEMBL11755946 0.86 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDLMNASLC22A1
SCHEMBL1543751 0.85 CDK1 (0.62) ALDH1A1KDM4EHPGDLMNASLC22A1
SCHEMBL7813262 0.84 RECQL (0.68) ALDH1A1LMNANOS2POLBTHRB
SCHEMBL22447558 0.84 ALDH1A1 (0.67) ALDH1A1KDM4EHPGDLMNASLC22A1
Hydrochloric Acid SCHEMBL9144741 0.84 CDK1 (0.60) ALDH1A1KDM4EHPGDLMNASLC22A1
SCHEMBL9410278 0.83 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDLMNASLC22A1
SCHEMBL10533123 0.81 ALDH1A1 (0.59) ALDH1A1KDM4EHPGDLMNASLC22A1
SCHEMBL11689255 0.81 NOS2 (0.63) ALDH1A1HPGDLMNACYP1A2CYP2C19
SCHEMBL11374040 0.80 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDLMNASLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620218-B1 2, 3-Dihydro-4(1H)-quinazolinones active in gastro-intestinal pathologies ALFA WASSERMANN SPA (IT) 1997-10-01 EP disclosed
US-5446152-A Antiemetic agent ALFA WASSERMANN S.P.A. (IT) 1995-08-29 US disclosed
EP-0620218-A1 Heterocyclic compounds active in gastro-intestinal pathologies ALFA WASSERMANN S.p.A. (IT) 1994-10-19 EP disclosed