SCHEMBL8771665

SCHEMBL8771665

CCOC(=O)c1ccc(N)cc1[N+](=O)[O-]

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.53
CYP3A4 P08684 3/20 0.53
TSHR P16473 2/20 0.53
RECQL P46063 1/20 0.53
NPC1 O15118 3/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
LMNA P02545 4/20 0.52
POLB P06746 3/20 0.52
GALR2 O43603 1/20 0.52
MITF O75030 1/20 0.52
HSP90AA1 P07900 1/20 0.52
HPGD P15428 1/20 0.52
XBP1 P17861 1/20 0.52
CCR6 P51684 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
ALOX15 P16050 3/20 0.49
HSD17B10 Q99714 3/20 0.49
CYP1A2 P05177 1/20 0.49
MAOA P21397 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16529634 0.85 ALDH1A1 (0.55) ALDH1A1CYP3A4TSHRNPC1SMN1; SMN2
SCHEMBL6422578 0.84 KMT2A (0.65) ALDH1A1NPC1SMN1; SMN2LMNAPOLB
SCHEMBL6750268 0.84 SMN1; SMN2 (0.65) ALDH1A1NPC1SMN1; SMN2LMNAPOLB
SCHEMBL2126420 0.84 CA12 (0.62) ALDH1A1TSHRNPC1SMN1; SMN2LMNA
SCHEMBL616603 0.83 GAA (0.63) ALDH1A1CYP3A4TSHRRECQLSMN1; SMN2
SCHEMBL31391703 0.82 MAPT (0.55) ALDH1A1TSHRNPC1SMN1; SMN2LMNA
SCHEMBL28999592 0.82 SMN1; SMN2 (0.53) ALDH1A1TSHRNPC1SMN1; SMN2LMNA
SCHEMBL6350616 0.82 ALDH1A1 (0.52) ALDH1A1TSHRNPC1SMN1; SMN2LMNA
SCHEMBL3092769 0.82 MAPT (0.55) ALDH1A1TSHRNPC1SMN1; SMN2LMNA
SCHEMBL29091595 0.81 MAPT (0.55) ALDH1A1NPC1SMN1; SMN2LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661259-B1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL MYERS SQUIBB CO (US) 1997-10-08 EP disclosed
US-5648385-A TREATING RHEUMATOID ARTHRITIS BRISTOL-MYERS SQUIBB CO. (US) 1997-07-15 US disclosed
US-5618839-A Retinoid-like compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-08 US disclosed
EP-0661259-A1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL-MYERS SQUIBB COMPANY (US) 1995-07-05 EP disclosed