SCHEMBL877233

SCHEMBL877233

Cc1c(Cc2ccc(OC(C)C)cc2)c(OC2OC(COC(=O)OCC3OC(Oc4nn(C(C)C)c(C)c4Cc4ccc(OC(C)C)cc4)C(O)C(O)C3O)C(O)C(O)C2O)nn1C(C)C

nearest known ligand 0.95

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SLC5A2 P31639 20/20 0.95
SLC5A1 P13866 18/20 0.95

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14634764 1.00 SLC5A2 (0.95) SLC5A2SLC5A1
SCHEMBL14634761 1.00 SLC5A2 (0.95) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL18432846 0.98 SLC5A2 (1.00) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL10066609 0.98 SLC5A2 (1.00) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL16421581 0.98 SLC5A2 (1.00) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL23072082 0.98 SLC5A2 (1.00) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL15168697 0.98 SLC5A2 (1.00) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL17034638 0.98 SLC5A2 (1.00) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL721678 0.98 SLC5A2 (1.00) SLC5A2SLC5A1
Remogliflozin Etabonate SCHEMBL10081649 0.98 SLC5A2 (1.00) SLC5A2SLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619198-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO Arena Pharmaceuticals, Inc. (US) 2013-07-31 EP claimed
EP-2556056-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO Arena Pharmaceuticals, Inc. (US) 2013-02-13 EP claimed
WO-2012040279-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2012-03-29 WO claimed
EP-2619198-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO Arena Pharmaceuticals, Inc. (US) 2013-07-31 EP disclosed
EP-2611427-A2 MODIFIED-RELEASE DOSAGE FORMS OF 5-HT2C AGONISTS USEFUL FOR WEIGHT MANAGEMENT& xA; Arena Pharmaceuticals, Inc. (US) 2013-07-10 EP disclosed
EP-2611782-A1 SALTS OF LORCASERIN WITH OPTICALLY ACTIVE ACIDS Arena Pharmaceuticals, Inc. (US) 2013-07-10 EP disclosed
EP-2611433-A2 NON-HYGROSCOPIC SALTS OF 5-HT2C AGONISTS Arena Pharmaceuticals, Inc. (US) 2013-07-10 EP disclosed
EP-2611781-A1 FAST-DISSOLVE DOSAGE FORMS OF 5-HT2C AGONISTS Arena Pharmaceuticals, Inc. (US) 2013-07-10 EP disclosed
WO-2013055910-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2013-04-18 WO disclosed
EP-2556056-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO Arena Pharmaceuticals, Inc. (US) 2013-02-13 EP disclosed
WO-2012170702-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2012-12-13 WO disclosed
WO-2012145361-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2012-10-26 WO disclosed
WO-2012145604-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2012-10-26 WO disclosed
WO-2012145603-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2012-10-26 WO disclosed
WO-2012135570-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2012-10-04 WO disclosed
WO-2012040279-A1 MODULATORS OF THE GPR119 RECEPTOR AND THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2012-03-29 WO disclosed
WO-2012030951-A1 FAST-DISSOLVE DOSAGE FORMS OF 5-HT2C AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2012-03-08 WO disclosed
WO-2012030957-A2 NON-HYGROSCOPIC SALTS OF 5-HT2C AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2012-03-08 WO disclosed
WO-2012030927-A2 MODIFIED-RELEASE DOSAGE FORMS OF 5-HT2C AGONISTS USEFUL FOR WEIGHT MANAGEMENT ARENA PHARMACEUTICALS, INC. (US) 2012-03-08 WO disclosed
WO-2012030938-A1 SALTS OF LORCASERIN WITH OPTICALLY ACTIVE ACIDS ARENA PHARMACEUTICALS, INC. (US) 2012-03-08 WO disclosed