SCHEMBL8772573

SCHEMBL8772573

C=CCc1cc(C(=O)OC(C)C)ccc1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.60
CA1 P00915 5/20 0.60
CA2 P00918 5/20 0.60
CA7 P43166 5/20 0.60
CA9 Q16790 5/20 0.60
CA14 Q9ULX7 5/20 0.60
HTT P42858 3/20 0.51
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
LMNA P02545 1/20 0.51
HSP90AA1 P07900 1/20 0.51
GABRA1 P14867 1/20 0.49
GABRB2 P47870 1/20 0.49
POLB P06746 1/20 0.47
PTPN1 P18031 4/20 0.46
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP4F2 P78329 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL542210 0.84 CA1 (0.57) CA12CA1CA2CA7CA9
SCHEMBL12088394 0.82 GAA (0.59) HTTALDH1A1HPGDLMNAHSP90AA1
SCHEMBL1515872 0.81 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL8772579 0.80 HTT (0.51) CA12CA1CA2CA9CA14
SCHEMBL1092424 0.79 HTT (0.71) HTTALDH1A1HPGDLMNAGABRA1
SCHEMBL8465492 0.78 HTT (0.61) CA12CA1CA2CA7CA9
SCHEMBL4943834 0.78 HTT (0.61) HTTALDH1A1HPGDLMNAGABRA1
SCHEMBL8419839 0.78 HDAC6 (0.50) CA12CA1CA2CA7CA9
SCHEMBL9550443 0.77 HTT (0.60) CA12CA1CA2CA7CA9
SCHEMBL39248 0.76 CA12 (1.00) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691349-A ANTICHOLESTEROL AGENTS; ATHEROSCLEROSIS ZENECA LIMITED (GB) 1997-11-25 US disclosed
EP-0654032-B1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LTD (GB) 1997-10-15 EP disclosed
EP-0654032-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS. ZENECA LTD (GB) 1995-05-24 EP disclosed
WO-1994003451-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1994-02-17 WO disclosed