SCHEMBL8772575

SCHEMBL8772575

CC1(C)CC=C(Sc2ccccc2)c2cc(C#Cc3ccc(C(=O)O)cc3)ccc21

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RARA P10276 19/20 0.68
RARB P10826 19/20 0.68
RARG P13631 19/20 0.68
CYP26A1 O43174 1/20 0.52
CYP3A4 P08684 1/20 0.52
CRABP2 P29373 1/20 0.52
RXRA P19793 1/20 0.47
NR2E1 Q9Y466 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6292573 0.87 RARB (0.50) RARARARBRARGRXRANR2E1
SCHEMBL8772596 0.87 RARA (0.52) RARARARBRARGCYP26A1CYP3A4
SCHEMBL8901315 0.84 RARA (0.64) RARARARBRARGCYP26A1CYP3A4
SCHEMBL8901265 0.83 RARB (0.63) RARARARBRARGCYP26A1CYP3A4
SCHEMBL8772545 0.83 RARB (0.63) RARARARBRARGCYP26A1CYP3A4
SCHEMBL6294021 0.83 RARA (0.69) RARARARBRARGRXRANR2E1
SCHEMBL6294022 0.83 RARA (0.69) RARARARBRARGRXRANR2E1
SCHEMBL7806999 0.82 RARA (0.78) RARARARBRARGCYP26A1CYP3A4
SCHEMBL6294125 0.82 HPGD (0.47) RARARARBRARGRXRANR2E1
SCHEMBL6210444 0.81 RARA (1.00) RARARARBRARGRXRANR2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed
US-5618931-A SKIN DISORDERS, ANTIINFLAMMATORY AGENTS ALLERGAN 1997-04-08 US disclosed
WO-1996020930-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-07-11 WO disclosed