SCHEMBL8772596

SCHEMBL8772596

CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(Sc2ccccc2)=CCC3(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARA P10276 19/20 0.52
RARB P10826 18/20 0.52
RARG P13631 18/20 0.52
CYP3A4 P08684 2/20 0.40
KMT2A Q03164 1/20 0.40
CYP26A1 O43174 1/20 0.39
CRABP2 P29373 1/20 0.39
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772575 0.87 RARA (0.68) RARARARBRARGCYP3A4CYP26A1
SCHEMBL8772557 0.87 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL8772538 0.86 RARA (0.52) RARARARBRARGCYP3A4KMT2A
SCHEMBL6423614 0.85 RARA (0.49) RARARARBRARGKMT2ATP53
SCHEMBL8915310 0.85 RARA (0.50) RARARARBRARGCYP3A4KMT2A
SCHEMBL7805699 0.84 RARA (0.60) RARARARBRARGCYP3A4KMT2A
SCHEMBL6240831 0.83 RARA (0.76) RARARARBRARG
SCHEMBL6451770 0.83 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL8915318 0.83 RARA (0.48) RARARARBRARGCYP3A4KMT2A
SCHEMBL7641992 0.83 RARA (0.56) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed
US-5618931-A SKIN DISORDERS, ANTIINFLAMMATORY AGENTS ALLERGAN 1997-04-08 US disclosed
WO-1996020930-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-07-11 WO disclosed