SCHEMBL8772728

SCHEMBL8772728

CCC(CC)=C1CCC(C)(C)c2cc(C#Cc3ccc(C(=O)O)cc3)ccc21

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RARB P10826 19/20 0.60
RARG P13631 19/20 0.60
RARA P10276 16/20 0.60
CYP26A1 O43174 2/20 0.60
CYP3A4 P08684 2/20 0.60
CRABP2 P29373 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8836860 0.91 RARB (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8836693 0.87 RARB (0.49) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7642401 0.82 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8836607 0.79 CYP26A1 (0.32) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8772525 0.78 RARB (0.47) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8836562 0.77 RARB (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL3302926 0.76 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL29353973 0.76 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7640552 0.75 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7642223 0.72 RARA (0.61) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed
US-5591858-A Acetylenes disubstituted with a 5 substituted tetrahydronaphthyl group and with an aryl or heteroaryl group having retinoid-like biological activity ALLERGAN 1997-01-07 US disclosed
WO-1996020930-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-07-11 WO disclosed
US-5514825-A SYNTHETIC RETINOIDS ALLERGAN, INC. (US) 1996-05-07 US disclosed