SCHEMBL8772863

SCHEMBL8772863

CSC(=NC#N)Nc1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.44
MAPT P10636 6/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
HTT P42858 4/20 0.44
TSHR P16473 2/20 0.44
LMNA P02545 2/20 0.44
NLRP3 Q96P20 1/20 0.44
IDO1 P14902 1/20 0.41
GAA P10253 2/20 0.41
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
PKM P14618 1/20 0.39
MAPK1 P28482 1/20 0.39
NPC1 O15118 4/20 0.39
RAB9A P51151 3/20 0.39
PTGIR P43119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15543683 0.85 MAPT (0.38) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL15543685 0.85 MAPT (0.38) ALDH1A1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL19069839 0.84 ALDH1A1 (0.41) ALDH1A1MAPTCYP1A2CYP2C19HTT
SCHEMBL10452571 0.83 NPC1 (0.50) ALDH1A1MAPTHTTTSHRLMNA
SCHEMBL10452569 0.83 NPC1 (0.50) ALDH1A1MAPTHTTTSHRLMNA
SCHEMBL10341391 0.83 ABCC9 (0.45) ALDH1A1MAPTHTTTSHRLMNA
SCHEMBL4104086 0.83 ALDH1A1 (0.43) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL4535023 0.83 ABCC9 (0.41) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL17402949 0.83 ABCC9 (0.41) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL4092695 0.83 ALDH1A1 (0.43) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625967-B1 N,N'-SUBSTITUTED IMIDOCARBONIMIDIC DIAMIDES DERIVED FROM HYDROXYLAMINES JACOBUS PHARMA CO INC (US) 1997-08-27 EP disclosed
US-5322858-A Antimicrobial, antiparasitic agents JACOBUS PHARMACEUTICAL CO. INC. (US) 1994-06-21 US disclosed
WO-1993016037-A1 N,N'-SUBSTITUTED IMIDOCARBONIMIDIC DIAMIDES DERIVED FROM HYDROXYLAMINES JACOBUS PHARMACEUTICAL CO., INC. (US) 1993-08-19 WO disclosed