SCHEMBL8773347

SCHEMBL8773347

C=CCN1CCN(CC=C)C(=O)N(CC=C)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.39
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
OPRD1 P41143 2/20 0.36
ADRA2A P08913 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
HRH3 Q9Y5N1 2/20 0.34
DRD2 P14416 2/20 0.34
MAPT P10636 2/20 0.34
ADRA1A P35348 2/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
DRD3 P35462 1/20 0.34
OPRK1 P41145 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL462082 0.91 CYP3A4 (0.46) CYP3A4LMNAGAAOPRD1MAPT
SCHEMBL9676287 0.83 CYP3A4 (0.39) CYP3A4
SCHEMBL20599288 0.82 CYP3A4 (0.42) CYP3A4LMNAGAAOPRD1OPRK1
SCHEMBL27797024 0.81 CYP3A4 (0.38) CYP3A4LMNAMAPTALDH1A1
SCHEMBL31469053 0.80 CYP3A4 (0.41) CYP3A4LMNAGAAADRA1AALDH1A1
SCHEMBL2871678 0.79 CYP3A4 (0.37) CYP3A4LMNAGAAALDH1A1
SCHEMBL9627129 0.79 HDAC3 (0.37) CYP3A4NPC1RAB9ALMNAGAA
SCHEMBL6692977 0.78 OPRD1 (0.41) CYP3A4NPC1RAB9ALMNAOPRD1
SCHEMBL290880 0.78
SCHEMBL327601 0.78 OPRD1 (0.41) CYP3A4NPC1RAB9ALMNAOPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670316-B1 1,3,6-Trialkylhexahydro-1,3,6-triazocine-2-one and preparation process thereof MITSUI TOATSU CHEMICALS (JP) 1997-09-03 EP claimed
JP-7291949-A None JP disclosed
JP-H07291949-A 1,3,6-TRIALKYLHEXAHYDRO-1,3,6-TRIAZOCIN-2-ONE AND PRODUCTION THEREOF MITSUI TOATSU CHEM INC 1995-11-07 JP disclosed