SCHEMBL8773415

SCHEMBL8773415

O=S(=O)(O)c1ccc(P(c2ccccc2)c2ccccc2)cc1.[NaH]

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
CYP2D6 P10635 2/20 0.53
POLB P06746 1/20 0.53
TDP1 Q9NUW8 3/20 0.52
CYP3A4 P08684 1/20 0.52
ESR1 P03372 2/20 0.52
ESR2 Q92731 2/20 0.52
LMNA P02545 1/20 0.48
ALDH1A1 P00352 4/20 0.46
NT5E P21589 1/20 0.46
SNCA P37840 1/20 0.41
MAPK1 P28482 1/20 0.38
HTR6 P50406 1/20 0.37
HSD17B10 Q99714 2/20 0.36
PTPRA P18433 1/20 0.36
PTPRB P23467 1/20 0.36
NAPRT Q6XQN6 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8145540 1.00 TSHR (0.62) TSHRSMN1; SMN2CYP2D6POLBTDP1
SCHEMBL996850 0.98 TSHR (0.65) TSHRSMN1; SMN2CYP2D6POLBTDP1
SCHEMBL718256 0.98 TSHR (0.65) TSHRSMN1; SMN2CYP2D6POLBTDP1
Water SCHEMBL570669 0.96 TSHR (0.62) TSHRSMN1; SMN2CYP2D6POLBTDP1
Water SCHEMBL30394765 0.96 TSHR (0.62) TSHRSMN1; SMN2CYP2D6POLBTDP1
Potassium SCHEMBL1450612 0.96 TSHR (0.62) TSHRSMN1; SMN2CYP2D6POLBTDP1
SCHEMBL6568428 0.96 TSHR (0.62) TSHRSMN1; SMN2CYP2D6POLBTDP1
SCHEMBL301148 0.96 TSHR (0.62) TSHRSMN1; SMN2CYP2D6POLBTDP1
SCHEMBL6569261 0.96 TSHR (0.62) TSHRSMN1; SMN2CYP2D6POLBTDP1
Water SCHEMBL1536886 0.94 TSHR (0.60) TSHRSMN1; SMN2CYP2D6POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5149868-A Carbonylation process SHELL OIL COMPANY (US) 1992-09-22 US claimed
US-20240216521-A1 METHODS OF PREPARING CELL-BINDING AGENT-DRUG CONJUGATES IMMUNOGEN INC (US) 2024-07-04 US disclosed
US-11833214-B2 Methods of preparing cell-binding agent-drug conjugates IMMUNOGEN, INC. (US) 2023-12-05 US disclosed
CN-110359097-B Method for obtaining On-DNA aromatic hydrocarbon compound through Suzuki coupling reaction in construction of DNA coding compound library 上海药明康德新药开发有限公司 2022-09-20 CN disclosed
CN-110331447-B Method for preparing On-DNA aryl alkyne compound in construction of DNA coding compound library 上海药明康德新药开发有限公司 2022-05-27 CN disclosed
EP-3941527-A1 METHODS OF PREPARING CELL-BINDING AGENT-DRUG CONJUGATES ImmunoGen, Inc. (US) 2022-01-26 EP disclosed
US-20200405874-A1 METHODS OF PREPARING CELL-BINDING AGENT-DRUG CONJUGATES IMMUNOGEN, INC. 2020-12-31 US disclosed
WO-2020191306-A1 METHODS OF PREPARING CELL-BINDING AGENT-DRUG CONJUGATES IMMUNOGEN, INC. (US) 2020-09-24 WO disclosed
EP-0489472-B1 Carbonylation process and catalyst composition SHELL INT RESEARCH (NL) 1997-10-29 EP disclosed
US-5149868-A Carbonylation process SHELL OIL COMPANY (US) 1992-09-22 US disclosed
EP-0489472-A2 Carbonylation process and catalyst composition SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1992-06-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11833214-B2 Methods of preparing cell-binding agent-drug conjugates EPCAM, CD2BP2, XPA TSHR 2222/4885SMN1; SMN2 3191/4885CYP2D6 2255/4885
US-20200405874-A1 METHODS OF PREPARING CELL-BINDING AGENT-DRUG CONJUGATES EPCAM, CD2BP2, XPA TSHR 2222/4885SMN1; SMN2 3191/4885CYP2D6 2255/4885
US-20240216521-A1 METHODS OF PREPARING CELL-BINDING AGENT-DRUG CONJUGATES EPCAM, CD2BP2, XPA TSHR 2222/4885SMN1; SMN2 3191/4885CYP2D6 2255/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.