SCHEMBL8774107

SCHEMBL8774107

CCCCC1CCC(CCc2ccc(-c3cc(F)c(F)nc3F)cc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.38
MAOB P27338 3/20 0.36
MAOA P21397 2/20 0.36
RARB P10826 3/20 0.36
HRH3 Q9Y5N1 1/20 0.36
FFAR4 Q5NUL3 1/20 0.33
RARA P10276 1/20 0.33
RARG P13631 1/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 2/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
S1PR1 P21453 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
S1PR3 Q99500 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774103 1.00 GPR84 (0.38) GPR84MAOBMAOARARBHRH3
SCHEMBL8774053 0.96 RARB (0.38) GPR84MAOBMAOARARBHRH3
SCHEMBL8774058 0.96 RARB (0.38) GPR84MAOBMAOARARBHRH3
SCHEMBL8775034 0.95 RARB (0.40) GPR84MAOBMAOARARBFFAR4
SCHEMBL8775036 0.95 RARB (0.40) GPR84MAOBMAOARARBFFAR4
SCHEMBL8774417 0.93 MAOB (0.38) GPR84MAOBMAOARARBHRH3
SCHEMBL8774424 0.93 MAOB (0.38) GPR84MAOBMAOARARBHRH3
SCHEMBL8774623 0.90 GPR84 (0.36) GPR84MAOBMAOAFFAR4
SCHEMBL8774619 0.90 GPR84 (0.36) GPR84MAOBMAOAFFAR4
SCHEMBL8775089 0.90 GPR84 (0.36) GPR84MAOBMAOARARBHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed