SCHEMBL8775188

SCHEMBL8775188

CC(=O)S.CCN(CC)CC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.42
CHRM4 P08173 2/20 0.42
CHRM5 P08912 2/20 0.42
CHRM1 P11229 2/20 0.42
CHRM3 P20309 2/20 0.42
ALDH1A1 P00352 5/20 0.40
HSD17B10 Q99714 2/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
TRPA1 O75762 1/20 0.37
ABCB11 O95342 1/20 0.36
CYP2E1 P05181 1/20 0.36
PTGS1 P23219 1/20 0.36
HTT P42858 1/20 0.36
GSDMD P57764 1/20 0.36
PAOX Q6QHF9 1/20 0.34
LMNA P02545 3/20 0.33
POLB P06746 1/20 0.32
CA12 O43570 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetone SCHEMBL3715272 0.86 LMNA (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5671517 0.84 ALDH1A1 (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetic Acid SCHEMBL28549045 0.83 FFAR3 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetic Acid SCHEMBL31218573 0.83 FFAR3 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetic Acid SCHEMBL28664565 0.83 FFAR3 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetic Acid SCHEMBL22152 0.83 FFAR3 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetic Acid SCHEMBL16244302 0.83 FFAR3 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetone SCHEMBL11644767 0.83 CHRM2 (0.44) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetic Acid SCHEMBL19356582 0.83 FFAR3 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
Acetic Acid SCHEMBL28289424 0.83 FFAR3 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805808-A1 PROCESS FOR THE PREPARATION OF 1-(THIOMETHYL)-CYCLOPROPANEACETIC ACID Merck & Co., Inc. (US) 1997-11-12 EP disclosed
WO-1996022987-A1 PROCESS FOR THE PREPARATION OF 1-(THIOMETHYL)-CYCLOPROPANEACETIC ACID MERCK & CO., INC. (US) 1996-08-01 WO disclosed
US-5523477-A REACTING 1,1-CYCLOPROPANEDIMETHANOL WITH DIALKYL SULFITE IN PRESENCE OF ACID OR BASE TO FORM CYCLIC SULFITE, REMOVING ALCOHOL REACTION BY-PRODUCT MERCK & CO., INC. (US) 1996-06-04 US disclosed