SCHEMBL8775412

SCHEMBL8775412

CCCCC/C(=C(/C)C(N)=O)N(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
CES2 O00748 4/20 0.41
CES1 P23141 4/20 0.41
FAAH O00519 3/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
AKR1B1 P15121 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
SOAT1 P35610 1/20 0.40
THRB P10828 1/20 0.40
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
PGGT1B P53609 1/20 0.40
PPARG P37231 6/20 0.39
PPARD Q03181 6/20 0.39
PPARA Q07869 6/20 0.39
GPR84 Q9NQS5 5/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28377249 1.00 ALDH1A1 (0.42) ALDH1A1CES2CES1FAAHMEN1
SCHEMBL8775139 0.98 CES2 (0.43) ALDH1A1CES2CES1FAAHMEN1
SCHEMBL27350149 0.98 CES2 (0.43) ALDH1A1CES2CES1FAAHMEN1
SCHEMBL27436232 0.94 ALDH1A1 (0.48) ALDH1A1CES2CES1FAAHMEN1
SCHEMBL2501493 0.94 ALDH1A1 (0.48) ALDH1A1CES2CES1FAAHMEN1
SCHEMBL33996 0.86 ALDH1A1 (0.37) ALDH1A1CES2CES1TSHR
SCHEMBL151388 0.86 ALDH1A1 (0.37) ALDH1A1CES2CES1TSHR
Hydrochloric Acid SCHEMBL5665875 0.84 ALDH1A1 (0.35) ALDH1A1CES2CES1TSHR
Hydrochloric Acid SCHEMBL14237669 0.84 ALDH1A1 (0.35) ALDH1A1CES2CES1TSHR
SCHEMBL9321835 0.82 FNTA (0.55) ALDH1A1CES2CES1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0606742-B1 Bile acid sequestrant ROHM & HAAS (US) 1997-11-19 EP claimed
US-5451397-A Crosslinked amino functional acrylic amide polymer, reducing blood cholesterol levels ROHM AND HAAS COMPANY (US) 1995-09-19 US claimed
EP-0606742-A1 Bile acid sequestrant ROHM AND HAAS COMPANY (US) 1994-07-20 EP claimed
EP-0606742-B1 Bile acid sequestrant ROHM & HAAS (US) 1997-11-19 EP disclosed
US-5451397-A Crosslinked amino functional acrylic amide polymer, reducing blood cholesterol levels ROHM AND HAAS COMPANY (US) 1995-09-19 US disclosed
EP-0606742-A1 Bile acid sequestrant ROHM AND HAAS COMPANY (US) 1994-07-20 EP disclosed