SCHEMBL8775479

SCHEMBL8775479

CC(c1ccccc1)N1CC(O)C2(CC2)C1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.49
OPRL1 P41146 6/20 0.48
OPRM1 P35372 5/20 0.48
OPRD1 P41143 4/20 0.48
OPRK1 P41145 4/20 0.48
MC4R P32245 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HSD11B1 P28845 1/20 0.41
KMT2A Q03164 1/20 0.38
CCR5 P51681 1/20 0.36
KCNA3 P22001 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL374064 1.00 CYP2D6 (0.49) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL3187502 0.81 CYP2D6 (0.49) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL13483618 0.81 CYP2D6 (0.49) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL769832 0.79 CYP2D6 (0.46) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL9596277 0.78 CYP2D6 (0.61) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL48088 0.78 CYP2D6 (0.61) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL2916607 0.78 CYP2D6 (0.61) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL4187954 0.78 CYP2D6 (0.45) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL4182073 0.78 CYP2D6 (0.45) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL8775418 0.76 CHRM2 (0.46) CYP2D6OPRL1OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529688-B1 Azaspiro(n,m)alkanes and diazaspiro(n,m)-alkanes DAIICHI SEIYAKU CO (JP) 1997-11-12 EP disclosed
US-5508428-A Spiro compound DAIICHI PHAMACEUTICAL CO., LTD. (JP) 1996-04-16 US disclosed
EP-0357047-B1 Spiro compounds DAIICHI SEIYAKU CO (JP) 1993-11-03 EP disclosed