SCHEMBL8775559

SCHEMBL8775559

O=C(O)C1CN(C2CC2)c2cc(F)c(F)cc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.35
TSHR P16473 1/20 0.33
NOTUM Q6P988 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5570112 0.89 PDE4A (0.35) TOP2ANOTUM
SCHEMBL17775397 0.84 TOP2A (0.42) TOP2ANOTUM
SCHEMBL16329562 0.83 TOP2A (0.55) TOP2ATSHRGAA
SCHEMBL22015414 0.81 TOP2A (0.44) TOP2ANOTUM
SCHEMBL21894264 0.81 TOP2A (0.42) TOP2ANOTUM
SCHEMBL8775774 0.78 ALDH1A1 (0.32) POLB
SCHEMBL12737551 0.77 TOP2A (0.40) TOP2ANOTUM
SCHEMBL23515125 0.75 TOP2A (0.44) TOP2A
SCHEMBL13667098 0.75 XIAP (0.32) TOP2A
SCHEMBL13667063 0.75 TOP2A (0.32) TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529688-B1 Azaspiro(n,m)alkanes and diazaspiro(n,m)-alkanes DAIICHI SEIYAKU CO (JP) 1997-11-12 EP disclosed
US-5508428-A Spiro compound DAIICHI PHAMACEUTICAL CO., LTD. (JP) 1996-04-16 US disclosed
US-5286723-A Spiro compound DAIICHI SEIYAKU CO., LTD. 1994-02-15 US disclosed
EP-0357047-B1 Spiro compounds DAIICHI SEIYAKU CO (JP) 1993-11-03 EP disclosed
EP-0529688-A2 Azaspiro n,m alkanes and diazaspiro n,m -alkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1993-03-03 EP disclosed
EP-0357047-A1 Spiro compounds DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1990-03-07 EP disclosed