SCHEMBL8776191

SCHEMBL8776191

COc1ncc(-c2ccc(Br)cc2)c(-c2ccc(S(N)(=O)=O)cc2)c1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.43
CA9 Q16790 3/20 0.43
CA12 O43570 2/20 0.43
PTGS2 P35354 12/20 0.42
PTGS1 P23219 7/20 0.42
CA1 P00915 3/20 0.41
CA4 P22748 1/20 0.41
CA5A P35218 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
KIF11 P52732 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8776179 0.87 PTGS2 (0.45) CA2CA9CA12PTGS2PTGS1
SCHEMBL8051564 0.73 PTGS2 (0.44) CA2CA9CA12PTGS2PTGS1
SCHEMBL7779954 0.69 LRRK2 (0.60) CA2CA9CA12PTGS2PTGS1
SCHEMBL8092791 0.67 PTGS2 (0.47) CA2CA9CA12PTGS2PTGS1
SCHEMBL6726344 0.65 PTGS2 (0.64) CA2CA9CA12PTGS2PTGS1
SCHEMBL24968929 0.65 ULK1 (0.37)
SCHEMBL30851331 0.65 ULK1 (0.37)
SCHEMBL6726396 0.65 PTGS2 (0.72) CA2CA9CA12PTGS2PTGS1
SCHEMBL6725900 0.65 CA12 (0.55) CA2CA9CA12PTGS2PTGS1
SCHEMBL8654649 0.64 PTGS2 (0.58) PTGS2PTGS1KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808305-A1 3,4-DIARYL SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024585-A1 3,4-DIARYL SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed