SCHEMBL8776300

SCHEMBL8776300

O=C(CCCCC(=O)N1CCN(c2ccncc2)CC1)N1CC[CH]CC1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.61
LMNA P02545 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
ITGB3 P05106 7/20 0.61
ITGA2B P08514 7/20 0.61
CHRM1 P11229 1/20 0.56
HTR1A P08908 2/20 0.53
HTR7 P34969 2/20 0.53
MMP2 P08253 1/20 0.52
ESR1 P03372 1/20 0.51
HDAC1 Q13547 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
F10 P00742 1/20 0.48
GRM5 P41594 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16596173 0.84 ITGB3 (0.62) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL8776254 0.83 SMN1; SMN2 (0.51) ITGB3ITGA2BSMN1; SMN2
SCHEMBL13801421 0.81 MAPT (0.58) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL7368202 0.81 ITGB3 (0.67) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL6600563 0.81 MAPT (0.62) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL4377713 0.79 ITGB3 (0.54) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL7787428 0.79 ITGB3 (0.60) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL8543870 0.79 ITGB3 (0.53) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL7791914 0.78 ITGB3 (0.61) MAPTLMNANPSR1ITGB3ITGA2B
SCHEMBL7790343 0.77 ITGB3 (0.69) MAPTLMNANPSR1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808311-A2 NEW DERIVATIVES OF PYRIDIL PIPERAZINE OR PYRIDAZINYL PIPERAZYL, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1997-11-26 EP disclosed
WO-1996024581-A2 DERIVATIVES OF PYRIDIL PIPERAZINE OR PYRIDAZINYL PIPERAZYL, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1996-08-15 WO disclosed