SCHEMBL7368202

SCHEMBL7368202

O=C(O)CCC(=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.67
ITGA2B P08514 9/20 0.67
ALDH1A1 P00352 2/20 0.60
HPGD P15428 2/20 0.60
HSD17B10 Q99714 2/20 0.60
KDM4E B2RXH2 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
RECQL P46063 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
LMNA P02545 1/20 0.58
MAPT P10636 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
HTR1A P08908 1/20 0.54
HTR7 P34969 1/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
CHRM1 P11229 1/20 0.53
MMP2 P08253 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27786793 0.85 MAPT (0.78) ALDH1A1HPGDHSD17B10KDM4ECYP3A4
SCHEMBL7790344 0.85 ITGB3 (0.60) ITGB3ITGA2BALDH1A1HPGDHSD17B10
SCHEMBL13801421 0.84 MAPT (0.58) ITGB3ITGA2BSMN1; SMN2LMNAMAPT
SCHEMBL6600563 0.84 MAPT (0.62) ITGB3ITGA2BCYP3A4CYP2C9LMNA
SCHEMBL4383007 0.84 MAPT (0.58) ITGB3ITGA2BALDH1A1SMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL4376006 0.83 MAPT (0.57) ITGB3ITGA2BALDH1A1LMNAMAPT
SCHEMBL17859454 0.81 ALDH1A1 (0.64) ALDH1A1HPGDHSD17B10SMN1; SMN2LMNA
SCHEMBL10015690 0.81 ALDH1A1 (0.86) ALDH1A1HPGDHSD17B10SMN1; SMN2LMNA
SCHEMBL8776300 0.81 MAPT (0.61) ITGB3ITGA2BSMN1; SMN2LMNAMAPT
SCHEMBL7790352 0.80 ITGB3 (0.60) ITGB3ITGA2BALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242600-B1 ANTIISCHEMIC AGENTS, ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-05 US disclosed
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed