SCHEMBL8776705

SCHEMBL8776705

CCCCOc1nc(-c2ccccc2F)c(-c2ccc(S(C)(=O)=O)cc2)cc1CNC

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.62
PTGS1 P23219 7/20 0.62
SCD O00767 1/20 0.39
FADS1 O60427 1/20 0.39
DRD1 P21728 1/20 0.39
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8094216 0.88 PTGS2 (0.80) PTGS2PTGS1
SCHEMBL8776827 0.83 PTGS2 (0.56) PTGS2PTGS1SCDFADS1DRD1
SCHEMBL8086783 0.79 PTGS2 (0.67) PTGS2PTGS1
SCHEMBL8093124 0.77 PTGS2 (0.78) PTGS2PTGS1
SCHEMBL8093929 0.77 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8098732 0.76 PTGS2 (0.83) PTGS2PTGS1
SCHEMBL8095458 0.75 PTGS2 (0.81) PTGS2PTGS1
SCHEMBL8098733 0.75 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL8094071 0.74 PTGS2 (0.80) PTGS2PTGS1
SCHEMBL8086507 0.74 PTGS2 (0.76) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed