SCHEMBL8776847

SCHEMBL8776847

CCSc1ccc(-c2cc(C#N)c(Cl)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 12/20 0.52
CNR2 P34972 5/20 0.52
CYP1A2 P05177 3/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
KDM1A O60341 1/20 0.41
CYP3A4 P08684 1/20 0.39
HPGD P15428 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093828 0.87 CNR1 (0.52) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL8776749 0.81 PTGS2 (0.47) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL2932218 0.80 CNR1 (0.49) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL8087025 0.78 PTGS2 (0.54)
SCHEMBL19835709 0.75 CNR1 (0.55) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL8100978 0.73 CNR1 (0.47) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL8085631 0.73 CNR1 (0.52) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL13498508 0.72 NPSR1 (0.69) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL2932221 0.72 RPS6KA3 (0.40) CNR1CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL5904231 0.72 CNR1 (0.56) CNR1CNR2CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed