SCHEMBL8776749

SCHEMBL8776749

CCS(=O)(=O)c1ccc(-c2cc(C#N)c(Cl)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.47
RORC P51449 1/20 0.43
PTGS1 P23219 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CNR1 P21554 8/20 0.41
CNR2 P34972 4/20 0.41
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8087025 0.88 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8776720 0.84 PTGS2 (0.47) PTGS2PTGS1NPSR1CNR1CNR2
SCHEMBL8776825 0.84 PTGS2 (0.46) PTGS2RORCPTGS1CNR1CNR2
SCHEMBL8776847 0.81 CNR1 (0.52) CYP1A2CYP2C9CYP2C19NPSR1CNR1
SCHEMBL8776822 0.79 PTGS2 (0.56) PTGS2PTGS1NPSR1CNR1CNR2
SCHEMBL2932218 0.79 CNR1 (0.49) CYP1A2CYP2C9CYP2C19NPSR1CNR1
SCHEMBL8093828 0.79 CNR1 (0.52) PTGS1CYP1A2CYP2C9CYP2C19NPSR1
SCHEMBL8776895 0.78 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL8776719 0.78 PTGS2 (0.44) PTGS2RORCPTGS1NPSR1CNR1
SCHEMBL8776742 0.77 PTGS2 (0.54) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed