SCHEMBL8777330

SCHEMBL8777330

CC(C)(C)OC(=O)CN(CCN(CCN(CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C)CC(=O)OCCCc1ccccc1)CC(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.48
CTDSP1 Q9GZU7 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
APOBEC3A P31941 2/20 0.45
APOBEC3G Q9HC16 2/20 0.45
MAPT P10636 1/20 0.45
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA4 P22748 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
NPC1 O15118 1/20 0.44
RECQL P46063 1/20 0.44
RAB9A P51151 1/20 0.44
CYP2D6 P10635 1/20 0.44
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
SCN1A P35498 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8886066 0.89 CA1 (0.58) CA1CA2CA4TDP1
SCHEMBL8777339 0.86 L3MBTL1 (0.54) CA1CA2CA4
SCHEMBL5557245 0.85 CA1 (0.51) ALDH1A1SMN1; SMN2CA1CA2CA4
SCHEMBL7737502 0.85 CA1 (0.51) ALDH1A1SMN1; SMN2CA1CA2CA4
SCHEMBL8874560 0.84 POLB (0.44) LMNAALDH1A1CA1CA2CA4
SCHEMBL19088163 0.84 LTA4H (0.42) ALDH1A1SMN1; SMN2TDP1MEN1KMT2A
SCHEMBL7562431 0.82 AKT1 (0.49) LMNACYP2D6MEN1KMT2ASCN1A
SCHEMBL23130693 0.81 AKT1 (0.50) LMNACYP2D6MEN1KMT2ASCN1A
SCHEMBL7570965 0.81 AKT1 (0.50) LMNACYP2D6MEN1KMT2ASCN1A
SCHEMBL30915258 0.81 AKT1 (0.50) LMNACYP2D6MEN1KMT2ASCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810990-A1 SUBSTITUTED DTPA MONOAMIDES OF CENTRAL CARBOXYLIC ACIDS AND METAL COMPLEXES THEREOF, PHARMACEUTICALS CONTAINING THESE COMPLEXES, DIAGNOSTIC AND THERAPEUTIC USES THEREOF AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1997-12-10 EP disclosed
US-5679852-A Process for the production of DTPA-monoamides of the central carboxylic acid and their use as pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-21 US disclosed
US-5676923-A SOLUBLE, STABLE, ORGAN-SPECIFIC NUCLEAR MAGNETIC RESONANCE CONTRAST AGENT SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-14 US disclosed
US-5676926-A Process for the production of DTPA-tetraesters of terminal carboxylic acids SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-14 US disclosed
WO-1996026182-A1 SUBSTITUTED DTPA MONOAMIDES OF CENTRAL CARBOXYLIC ACIDS AND METAL COMPLEXES THEREOF, PHARMACEUTICALS CONTAINING THESE COMPLEXES, DIAGNOSTIC AND THERAPEUTIC USES THEREOF AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1996-08-29 WO disclosed
US-5514810-A Process for the production of DTPA-tetraesters of terminal carboxylic acids SCHERING AKTIENGESELLSCHAFT (DE) 1996-05-07 US disclosed