SCHEMBL8778050

SCHEMBL8778050

CCOC(=O)CNC(=O)[C@H](CCSC)NC(=O)OC(C)(C)C

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.66
CTSS P25774 6/20 0.66
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
HTT P42858 1/20 0.52
CA2 P00918 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
EPHX2 P34913 1/20 0.42
HPGD P15428 1/20 0.42
BACE1 P56817 1/20 0.42
TSHR P16473 1/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL9787694 0.96 CTSK (0.62) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL7436235 0.88 CTSS (0.70) CTSKCTSSCA2ALDH1A1KDM4E
SCHEMBL3721596 0.88 CTSS (0.70) CTSKCTSSCA2ALDH1A1KDM4E
SCHEMBL10606387 0.88 CTSS (0.70) CTSKCTSSCA2ALDH1A1KDM4E
SCHEMBL19115973 0.87 CTSK (0.65) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL19709962 0.86 CYP1A2 (0.59) CTSKCTSSCYP1A2CYP2C9CYP2C19
SCHEMBL9611898 0.86 CTSS (0.74) CTSKCTSSCA2ALDH1A1KDM4E
SCHEMBL10606688 0.86 CTSS (0.74) CTSKCTSSCA2ALDH1A1KDM4E
SCHEMBL19709746 0.85 CYP1A2 (0.55) CTSKCTSSCYP1A2CYP2C9CYP2C19
Iodide SCHEMBL7508332 0.85 CTSS (0.66) CTSKCTSSCA2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802923-A1 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1997-10-29 EP disclosed
WO-1995035311-A1 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1995-12-28 WO disclosed
US-4997950-A Antisecretory MURPHY RICHARD FINBAR (US) 1991-03-05 US disclosed