SCHEMBL8779398

SCHEMBL8779398

Nc1nnc(SCc2ccc([N+](=O)[O-])cc2)s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.72
MAPT P10636 5/20 0.72
LMNA P02545 3/20 0.72
HTT P42858 3/20 0.71
TP53 P04637 1/20 0.71
RAB9A P51151 4/20 0.64
GAA P10253 4/20 0.64
LCK P06239 1/20 0.61
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60
MGAM O43451 1/20 0.56
SI P14410 1/20 0.56
MGAM2 Q2M2H8 1/20 0.56
NPC1 O15118 2/20 0.55
ABL1 P00519 3/20 0.54
SRC P12931 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.53
TSHR P16473 1/20 0.53
POLB P06746 1/20 0.51
GFER P55789 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16150878 0.86 LCK (0.61) ALDH1A1MAPTLMNAHTTTP53
SCHEMBL10532529 0.78 MAPT (0.58) ALDH1A1MAPTLMNAHTTTP53
SCHEMBL8177453 0.77 NPC1 (0.67) ALDH1A1HTTRAB9ANPC1ABL1
SCHEMBL8779332 0.77 NPC1 (0.63) ALDH1A1HTTRAB9AGAAMEN1
SCHEMBL8779275 0.77 NPC1 (0.62) ALDH1A1LMNAHTTRAB9AGAA
SCHEMBL3906094 0.77 MAPK1 (0.62) ALDH1A1MAPTLMNAHTTRAB9A
SCHEMBL10363026 0.77 MAPT (0.67) ALDH1A1MAPTLMNAHTTTP53
SCHEMBL8779378 0.76 ABL1 (0.70) ALDH1A1MAPTLMNAHTTTP53
SCHEMBL14426475 0.75 LMNA (0.74) ALDH1A1MAPTLMNAHTTRAB9A
SCHEMBL7481344 0.75 NPC1 (0.56) ALDH1A1HTTRAB9AGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579129-B1 Thiadiazole derivatives for the treatment of depressive states CT LAB FARM SRL (IT) 1997-03-05 EP claimed
EP-0579129-A2 Thiadiazole derivatives for the treatment of depressive states LABORATORIO FARMACEUTICO C.T. S.r.l. (IT) 1994-01-19 EP claimed