SCHEMBL8779983

SCHEMBL8779983

CS(=O)(=O)c1cccc(N2CCCCC2)c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.64
HTR6 P50406 3/20 0.53
GPR119 Q8TDV5 1/20 0.51
MLYCD O95822 1/20 0.48
NR1H2 P55055 5/20 0.48
NR1H3 Q13133 4/20 0.48
PTGS2 P35354 1/20 0.48
PRMT6 Q96LA8 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPT P10636 2/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13800992 0.98 DRD2 (0.66) DRD2HTR6GPR119MLYCDNR1H2
SCHEMBL21442594 0.85 DRD2 (0.71) DRD2HTR6GPR119MLYCDNR1H2
SCHEMBL17893525 0.83 DRD2 (0.61) DRD2HTR6GPR119MLYCDNR1H2
SCHEMBL3454087 0.83 HTR6 (0.70) DRD2HTR6
SCHEMBL23043686 0.83 HTR6 (0.58) DRD2HTR6MEN1ALDH1A1KMT2A
SCHEMBL29978549 0.83 HTR6 (0.58) DRD2HTR6MEN1ALDH1A1KMT2A
SCHEMBL17856468 0.83 CA1 (0.53) HTR6KDM4EMEN1ALDH1A1GAA
SCHEMBL12367089 0.82 DRD2 (0.59) DRD2HTR6GPR119MLYCDNR1H2
SCHEMBL38652751 0.81 CA1 (0.55) DRD2HTR6KDM4EMEN1ALDH1A1
SCHEMBL38652729 0.81 HTR6 (0.54) DRD2HTR6KDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100345833-C Modulators of dopamine neurotransmission CARLSSON RES AB (SE) 2007-10-31 CN disclosed
CN-1255382-C Novel modulators of dopamine neurotransmission CARLSSON A RESEARCH AB (SE) 2006-05-10 CN disclosed
CN-1765890-A Modulators of dopamine neurotransmission CARLSSON RES AB (SE) 2006-05-03 CN disclosed
CN-1420869-A Novel modulators of dopamine neurotransmission CARLSSON A RESEARCH AB (SE) 2003-05-28 CN disclosed
EP-0783486-A1 NOVEL PROSTAGLANDIN SYNTHASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-07-16 EP disclosed