SCHEMBL8780424

SCHEMBL8780424

CCCCC(Nc1ccccc1C(F)(F)F)=C(C(=O)O)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
POLB P06746 3/20 0.52
GAA P10253 3/20 0.52
MAPK1 P28482 1/20 0.51
EPHX2 P34913 1/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
HPGD P15428 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
KMT2A Q03164 4/20 0.47
MEN1 O00255 2/20 0.47
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 1/20 0.47
THRB P10828 1/20 0.47
RAB9A P51151 1/20 0.47
NOX1 Q9Y5S8 1/20 0.47
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780472 0.95 ALDH1A1 (0.52) ALDH1A1POLBGAAMAPK1EPHX2
SCHEMBL8780440 0.89 ALDH1A1 (0.50) ALDH1A1POLBGAAMAPK1EPHX2
SCHEMBL11619781 0.85 ALDH1A1 (0.53) ALDH1A1POLBGAAMAPK1EPHX2
SCHEMBL11616583 0.83 ALDH1A1 (0.67) ALDH1A1POLBGAAMAPK1CYP1A2
SCHEMBL11616203 0.83 ALDH1A1 (0.51) ALDH1A1POLBGAAMAPK1CYP1A2
SCHEMBL6017228 0.79 POLB (0.63) ALDH1A1POLBGAAMAPK1EPHX2
SCHEMBL11616199 0.78 ALDH1A1 (0.54) ALDH1A1POLBGAAMAPK1CYP1A2
SCHEMBL4145745 0.78 GAA (0.62) ALDH1A1POLBGAAEPHX2CYP1A2
SCHEMBL11617140 0.77 KMT2A (0.49) ALDH1A1POLBGAAMAPK1EPHX2
SCHEMBL11622880 0.77 POLB (0.54) ALDH1A1POLBGAAMAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP claimed
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP disclosed