SCHEMBL8780455

SCHEMBL8780455

NC(=O)/C=C1/CCCc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.56
NOTUM Q6P988 1/20 0.48
CYP19A1 P11511 5/20 0.47
CYP11B1 P15538 5/20 0.47
CYP11B2 P19099 5/20 0.47
MAPT P10636 4/20 0.47
MIF P14174 2/20 0.47
CYP2A6 P11509 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 1/20 0.47
TP53 P04637 1/20 0.47
NFKB1 P19838 1/20 0.47
RAB9A P51151 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780459 1.00 RXRA (0.56) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL9391471 0.89 CES1 (0.45) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL9391477 0.89 CES1 (0.45) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL9391470 0.89 CES1 (0.45) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL16168486 0.87 RXRA (0.45) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL8923628 0.84 RXRA (0.60) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL12629637 0.84 RXRA (0.60) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL8923632 0.84 RXRA (0.60) RXRANOTUMCYP19A1CYP11B1CYP11B2
SCHEMBL3253387 0.81 RXRA (0.60) RXRACYP19A1CYP11B1CYP11B2MAPT
SCHEMBL13545387 0.79 RXRA (0.52) RXRACYP19A1CYP11B1CYP11B2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759025-A1 AMIDE DERIVATIVES AND THEIR THERAPEUTIC USE THE WELLCOME FOUNDATION LIMITED (GB) 1997-02-26 EP disclosed
WO-1995030644-A1 AMIDE DERIVATIVES AND THEIR THERAPEUTIC USE THE WELLCOME FOUNDATION LIMITED (GB) 1995-11-16 WO disclosed