SCHEMBL8780925

SCHEMBL8780925

CN(CCOc1ccc(NS(C)(=O)=O)cc1)CCc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.65
CACNA1F O60840 1/20 0.65
CHRM2 P08172 1/20 0.65
ACHE P22303 1/20 0.65
AGTR1 P30556 1/20 0.65
DRD3 P35462 1/20 0.65
CACNA1D Q01668 1/20 0.65
CACNA1S Q13698 1/20 0.65
CACNA1C Q13936 1/20 0.65
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
LTA4H P09960 1/20 0.44
MAPK1 P28482 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 1/20 0.41
GRIN1 Q05586 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780850 0.94 KCNH2 (0.59) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780777 0.88 KCNH2 (0.48) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8781017 0.87 NPC1 (0.48) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780810 0.84 NPC1 (0.47) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780849 0.84 KCNH2 (0.47) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780917 0.83 NPC1 (0.49) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780876 0.82 NPC1 (0.48) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780867 0.82 KCNH2 (0.43) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780936 0.82 KCNH2 (0.54) KCNH2CACNA1FCHRM2ACHEAGTR1
Dofetilide SCHEMBL6102734 0.79 KCNH2 (1.00) KCNH2CACNA1FCHRM2ACHEAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed