SCHEMBL8780867

SCHEMBL8780867

CN(CCOc1ccc(N)cc1)CCc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.43
CACNA1F O60840 1/20 0.39
CHRM2 P08172 1/20 0.39
ACHE P22303 1/20 0.39
AGTR1 P30556 1/20 0.39
DRD3 P35462 1/20 0.39
CACNA1D Q01668 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
MCHR1 Q99705 2/20 0.39
PKM P14618 2/20 0.38
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
DRD2 P14416 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780990 0.93 KCNH2 (0.39) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780940 0.86 ADORA2A (0.43) KCNH2MCHR1PKMADORA3ADORA2A
SCHEMBL8780824 0.85 TDP1 (0.39) KCNH2MCHR1PKMADORA3ADORA2A
SCHEMBL8780815 0.85 ADORA2A (0.38) KCNH2ACHEMCHR1PKMADORA3
SCHEMBL8780872 0.84 KCNH2 (0.63) KCNH2PKMSIGMAR1HRH3SMN1; SMN2
SCHEMBL8780925 0.82 KCNH2 (0.65) KCNH2CACNA1FCHRM2ACHEAGTR1
SCHEMBL8780789 0.81 ADORA2A (0.41) KCNH2MCHR1PKMADORA3ADORA2A
SCHEMBL8780781 0.81 LTA4H (0.46) KCNH2MCHR1SMN1; SMN2
SCHEMBL8780750 0.81 TDP1 (0.37) KCNH2MCHR1PKMADORA3ADORA2A
SCHEMBL8780776 0.81 MAOA (0.37) KCNH2CHRM2ACHEDRD3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed