SCHEMBL8782006

SCHEMBL8782006

Cc1cc(F)ccc1OCc1ccccc1C(=O)C#N

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 5/20 0.49
SGMS2 Q8NHU3 1/20 0.43
FFAR4 Q5NUL3 5/20 0.42
FFAR1 O14842 3/20 0.42
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
PPARA Q07869 1/20 0.41
PTGDR2 Q9Y5Y4 2/20 0.41
FOLH1 Q04609 1/20 0.40
NOTUM Q6P988 1/20 0.40
MAPK14 Q16539 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8782060 0.88 MRGPRX4 (0.47) MRGPRX4FFAR4FFAR1FOLH1MAPT
SCHEMBL8101220 0.87 RXRA (0.47) SGMS2TP53HTTPTGDR2FOLH1
SCHEMBL8782034 0.85 MRGPRX4 (0.55) MRGPRX4FFAR4FFAR1TP53HTT
SCHEMBL8782322 0.84 FFAR4 (0.48) MRGPRX4FFAR4FFAR1FOLH1
SCHEMBL8782203 0.84 MRGPRX4 (0.52) MRGPRX4SGMS2FFAR4FFAR1TP53
Toluene SCHEMBL28735228 0.82 RXRA (0.46) MRGPRX4SGMS2TP53HTTPTGDR2
SCHEMBL8782015 0.82 HTT (0.47) MRGPRX4SGMS2TP53HTTFOLH1
SCHEMBL8783068 0.80 TP53 (0.48) MRGPRX4SGMS2TP53HTTPTGDR2
SCHEMBL8782268 0.80 NR4A2 (0.48) MRGPRX4MEN1KMT2A
SCHEMBL8782010 0.79 FFAR1 (0.46) FFAR4FFAR1TP53HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0718279-B1 Process for the preparation of o-substituted benzoylcyanides BASF AG (DE) 1997-09-24 EP disclosed
EP-0718279-A1 Process for the preparation of o-substituted benzoylcyanides BASF AKTIENGESELLSCHAFT (DE) 1996-06-26 EP disclosed
US-5221762-A Reacting a phenol with benzolactone compound; then phosgene or thionyl chloride; esterification with alcohol BASF AKTIENGESELLSCHAFT (DE) 1993-06-22 US disclosed
EP-0493711-A1 Process for the preparation of E-oximethers from phenylglyoxylic acid esters BASF Aktiengesellschaft (DE) 1992-07-08 EP disclosed