SCHEMBL8782015

SCHEMBL8782015

N#CC(=O)c1ccccc1COc1ccccc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.47
TP53 P04637 2/20 0.47
MRGPRX4 Q96LA9 2/20 0.44
NPC1 O15118 1/20 0.44
SGMS2 Q8NHU3 1/20 0.44
ALDH1A1 P00352 5/20 0.43
MCL1 Q07820 1/20 0.43
LMNA P02545 4/20 0.43
CXCL8 P10145 1/20 0.42
USP2 O75604 1/20 0.42
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
MAPT P10636 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
FOLH1 Q04609 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8783068 0.84 TP53 (0.48) HTTTP53MRGPRX4SGMS2ALDH1A1
SCHEMBL8782010 0.83 FFAR1 (0.46) HTTTP53ALDH1A1MEN1KMT2A
SCHEMBL8101220 0.83 RXRA (0.47) HTTTP53SGMS2ALDH1A1MAPT
SCHEMBL8782020 0.83 TP53 (0.69) HTTTP53MRGPRX4NPC1SGMS2
SCHEMBL9442060 0.82 RXRA (0.50) HTTTP53MRGPRX4SGMS2ALDH1A1
SCHEMBL8782006 0.82 MRGPRX4 (0.49) HTTTP53MRGPRX4SGMS2MEN1
SCHEMBL8782250 0.81 HTT (0.54) HTTTP53MRGPRX4NPC1SGMS2
SCHEMBL8594751 0.81 ALDH1A1 (0.46) HTTTP53MRGPRX4NPC1SGMS2
SCHEMBL8594755 0.81 ALDH1A1 (0.46) HTTTP53MRGPRX4NPC1SGMS2
SCHEMBL8069191 0.79 KDM4E (0.48) HTTTP53NPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0718279-B1 Process for the preparation of o-substituted benzoylcyanides BASF AG (DE) 1997-09-24 EP disclosed
EP-0718279-A1 Process for the preparation of o-substituted benzoylcyanides BASF AKTIENGESELLSCHAFT (DE) 1996-06-26 EP disclosed
US-5221762-A Reacting a phenol with benzolactone compound; then phosgene or thionyl chloride; esterification with alcohol BASF AKTIENGESELLSCHAFT (DE) 1993-06-22 US disclosed
EP-0493711-A1 Process for the preparation of E-oximethers from phenylglyoxylic acid esters BASF Aktiengesellschaft (DE) 1992-07-08 EP disclosed