SCHEMBL8783196

SCHEMBL8783196

CN1C(=O)c2ccccc2CC1c1ccc(O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.45
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
HTR2B P41595 2/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ESR2 Q92731 1/20 0.42
DRD2 P14416 2/20 0.41
DRD3 P35462 1/20 0.41
NPC1 O15118 1/20 0.40
CYP3A4 P08684 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
CAPN1 P07384 1/20 0.40
MAOB P27338 1/20 0.40
HTR1A P08908 1/20 0.39
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8782404 0.83 NPC1 (0.51) MEN1KMT2ADRD3NPC1MAPT
SCHEMBL8782099 0.83 HTR2A (0.44) HTR2AHTR2CHTR2BDRD2HTR1A
SCHEMBL8782066 0.81 KMT2A (0.49) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL3888787 0.76 KDM4E (0.53) KDM4EMEN1KMT2ACYP3A4MAPT
SCHEMBL9407110 0.76 PBRM1 (0.37) ESR1KDM4EMEN1KMT2AESR2
SCHEMBL8782123 0.75 DRD2 (0.46) ESR1MEN1KMT2AESR2DRD2
SCHEMBL28922579 0.74 HTR2C (0.49) HTR2AHTR2CHTR2BKDM4EKMT2A
SCHEMBL15041795 0.73 HTR2C (0.53) HTR2AHTR2CHTR2BKMT2ACAPN1
SCHEMBL10855534 0.71 CAPN1 (0.56) HTR2AHTR2CHTR2BKDM4ECAPN1
SCHEMBL8498408 0.71 CAPN1 (0.56) HTR2AHTR2CHTR2BKDM4ECAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0495610-B1 Tetrahydroisoquinoline derivatives, processes for producing the same and fungicides containing the same TOSOH CORP (JP) 1997-06-18 EP disclosed
US-5401752-A EFFECTIVE AGAINST DRUG RESISTANT FUNGI TOSOH CORPORATION (JP) 1995-03-28 US disclosed
EP-0495610-A1 Tetrahydroisoquinoline derivatives, processes for producing the same and fungicides containing the same TOSOH CORPORATION (JP) 1992-07-22 EP disclosed