SCHEMBL9407110

SCHEMBL9407110

CN1C(=O)c2cc(O)ccc2CC1c1ccc(C(C)(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.37
LMNA P02545 2/20 0.37
TYR P14679 1/20 0.37
RIPK1 Q13546 1/20 0.36
PRKCZ Q05513 2/20 0.36
CRBN Q96SW2 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
RGS12 O14924 1/20 0.36
CYP1A2 P05177 1/20 0.36
DRD2 P14416 1/20 0.36
PKM P14618 1/20 0.36
NFKB1 P19838 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428138 0.86 ACHE (0.41) RIPK1HDAC3HDAC1HDAC2HDAC8
SCHEMBL9427965 0.83 USP2 (0.36) RIPK1HDAC3HDAC1HDAC2HDAC8
SCHEMBL8782099 0.82 HTR2A (0.44) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL8783196 0.76 ESR1 (0.45) ESR1ESR2MAPTDRD2MAPK1
SCHEMBL9429146 0.69 HRH3 (0.36) RIPK1PRKCZHPGD
SCHEMBL9427669 0.66 TSHR (0.38) RIPK1PRKCZ
SCHEMBL7598342 0.66 AR (0.71) ESR1ESR2MAPTCYP1A2MAPK1
SCHEMBL29678628 0.65 PBRM1 (0.53) PBRM1CRBNDRD2KMT2AMEN1
SCHEMBL1037654 0.65 PBRM1 (0.53) PBRM1CRBNDRD2KMT2AMEN1
SCHEMBL8782370 0.64 DRD2 (0.39) RIPK1PRKCZHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-6211798-A None JP disclosed
JP-H06211798-A TETRAHYDROISOQUINOLINE DERIVATIVE AND ITS PRODUCTION TOSOH CORP 1994-08-02 JP disclosed