SCHEMBL8784228

SCHEMBL8784228

N#CCc1cccc(Oc2ccc(Cl)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
PPARG P37231 1/20 0.49
PPARA Q07869 1/20 0.49
LMNA P02545 1/20 0.49
FDFT1 P37268 2/20 0.43
AR P10275 2/20 0.43
ENPP2 Q13822 1/20 0.42
DAGLA Q9Y4D2 1/20 0.41
FFAR1 O14842 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
FAAH O00519 2/20 0.41
MMP3 P08254 1/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10547199 0.89 AR (0.48) ALDH1A1LMNAARENPP2FFAR1
SCHEMBL11034783 0.88 KDM4E (0.49) ALDH1A1PPARGPPARAENPP2FFAR1
SCHEMBL30641469 0.86 FFAR1 (0.47) ALDH1A1FDFT1ENPP2FFAR1FFAR4
SCHEMBL191669 0.86 FFAR1 (0.47) ALDH1A1FDFT1ENPP2FFAR1FFAR4
SCHEMBL10547112 0.86 KMO (0.51) ALDH1A1PPARGPPARAFDFT1ENPP2
SCHEMBL10547235 0.84 ALDH1A1 (0.51) ALDH1A1PPARGPPARALMNAFDFT1
SCHEMBL8597193 0.84 AR (0.50) ALDH1A1LMNAARMAPT
SCHEMBL10550577 0.84 FFAR4 (0.49) ALDH1A1FDFT1ENPP2FFAR1FFAR4
SCHEMBL10545623 0.84 SMN1; SMN2 (0.56) ALDH1A1ARENPP2
SCHEMBL8454764 0.84 NPSR1 (0.43) ALDH1A1ENPP2FFAR1FFAR4FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0595995-B1 ARYLAMIDOALKYL- AND ARYLAMINOALKYL-N-HYDROXYUREA COMPOUNDS AND -N-HYDROXYFORMAMIDE DERIVATIVES HAVING LIPOXYGENASE INHIBITORY ACTIVITY ABBOTT LAB (US) 1997-01-15 EP disclosed
US-5514702-A Arylamidoalkyl-N-hydroxyurea compounds having lipoxygenase inhibitory activity ABBOTT LABORATORIES (US) 1996-05-07 US disclosed
US-4814340-A 1,4-diaryl alkane derivatives having insecticidal and acaricidal activity MITSUI TOATSU CHEMICALS, INC. (JP) 1989-03-21 US disclosed
US-4661501-A Certain aryl-alkane-2-pyridyloxy-phenyl derivatives having insecticidal and acaricidal activity MITSUI TOATSU CHEMICALS, INC. (JP) 1987-04-28 US disclosed
EP-0091208-B1 METHOD FOR COMBATING INSECT PESTS, AND NOVEL CYCLOPROPANE CARBOXYLATES USEFUL AS ACTIVE INGREDIENTS THEREIN IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-06-18 EP disclosed
US-4532258-A Controlling insects, mites, pests KURARAY CO., LTD. (JP) 1985-07-30 US disclosed
EP-0091208-A1 Method for combating insect pests, and novel cyclopropane carboxylates useful as active ingredients therein IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-10-12 EP disclosed
US-4390547-A 2,2-Dimethyl-3-(substituted ethyl)cyclopropane carboxylate pesticidal compositions and methods KURARAY CO., LTD. (JP) 1983-06-28 US disclosed
US-4299839-A Novel pesticides and pesticidal compositions cyclopropanecarboxylates and pesticidal method KURARAY CO., LTD. (JP) 1981-11-10 US disclosed
US-4277490-A Insecticidal 1-(2-naphthyl)-cyclobutane carboxylate COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANIZATION (AU) 1981-07-07 US disclosed
EP-0002620-A1 Cycloalkyl carboxylic esters, insecticidal compositions containing them, and methods for their preparation COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1979-06-27 EP disclosed