SCHEMBL8784248

SCHEMBL8784248

CN1CCC(c2c[nH]c3ccc(-c4c[nH]nn4)cc23)C1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
ATM Q13315 1/20 0.57
HTR1D P28221 7/20 0.52
HTR1B P28222 7/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
THPO P40225 1/20 0.52
APP P05067 1/20 0.47
GABRP O00591 1/20 0.47
GABRD O14764 1/20 0.47
GABRA1 P14867 1/20 0.47
GABRB1 P18505 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRA2 P47869 1/20 0.47
GABRB2 P47870 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8784407 0.93 HTR1D (0.60) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL8097614 0.81 KDM4E (0.58) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8785321 0.80 HTR2C (0.52) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL2926854 0.79 KDM4E (0.67) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8090606 0.79 KDM4E (0.54) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8474262 0.79 KDM4E (0.56) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8508491 0.78 KDM4E (0.68) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8686333 0.77 KDM4E (0.57) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL25072243 0.77 MTNR1A (0.65) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL30877857 0.77 KDM4E (0.67) KDM4EATMHTR1DHTR1BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497512-B1 Imidazole, triazole and tetrazole derivatives MERCK SHARP & DOHME (GB) 1997-09-24 EP disclosed